SCHEMBL7449809

SCHEMBL7449809

O=C(N1CCCC1)C1(c2ccc3nc[nH]c3c2)CC1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 9/20 0.51
ALDH1A1 P00352 4/20 0.46
HPGD P15428 2/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
EPHX2 P34913 1/20 0.45
KDM4E B2RXH2 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
EPHX1 P07099 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
GPR183 P32249 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7449807 0.90 HSD11B1 (0.51) HSD11B1ALDH1A1HPGDMEN1KMT2A
SCHEMBL12431600 0.74 ALDH1A1 (0.71) HSD11B1ALDH1A1HPGDMEN1KMT2A
SCHEMBL4664222 0.73 EPHX2 (0.44) HSD11B1ALDH1A1HPGDEPHX2KDM4E
SCHEMBL1078194 0.73 RAF1 (0.40) HSD11B1ALDH1A1HPGDEPHX2KDM4E
SCHEMBL5805385 0.73 ALDH1A1 (0.70) HSD11B1ALDH1A1HPGDMEN1KMT2A
SCHEMBL2595556 0.72 EPHX2 (0.47) HSD11B1ALDH1A1HPGDEPHX2KDM4E
SCHEMBL1464875 0.70 AKR1C3 (0.41) ALDH1A1HPGDKDM4ESMN1; SMN2EPHX1
SCHEMBL5094333 0.70 HSD11B1 (0.67) HSD11B1ALDH1A1HPGDMEN1KMT2A
SCHEMBL17804163 0.69 HSD11B1 (0.66) HSD11B1ALDH1A1MEN1KMT2ALMNA
SCHEMBL348724 0.68 HSD11B1 (1.00) HSD11B1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095025-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-05-02 EP disclosed
WO-2000001704-A2 BENZIMIDAZOLES, PRODUCTION THEREOF AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-01-13 WO disclosed