SCHEMBL7450183

SCHEMBL7450183

CC(=O)c1ccc(C#N)cc1Br

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
TTR P02766 1/20 0.44
ALB P02768 1/20 0.44
CXCR1 P25024 1/20 0.40
CXCR2 P25025 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
GSK3B P49841 4/20 0.38
NCEH1 Q6PIU2 1/20 0.38
XDH P47989 1/20 0.37
SLC22A12 Q96S37 1/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
FFAR1 O14842 1/20 0.37
DYRK1A Q13627 1/20 0.37
PTPN1 P18031 2/20 0.36
PTPN2 P17706 1/20 0.36
LRRK2 Q5S007 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25255223 0.85 MEN1 (0.47) MEN1KMT2ATTRALBCXCR1
SCHEMBL23674669 0.83 XDH (0.49) MEN1KMT2ATTRALBCXCR1
SCHEMBL17109321 0.81 MEN1 (0.44) MEN1KMT2ATTRALBCXCR1
SCHEMBL28276264 0.81 CASP1 (0.44) MEN1KMT2ATTRALBCXCR1
SCHEMBL27839112 0.81 RAB9A (0.42) MEN1KMT2ATTRALBCXCR1
SCHEMBL4778338 0.81 CA12 (0.42) MEN1KMT2ATTRALBCXCR1
SCHEMBL8757233 0.79 SMN1; SMN2 (0.41) MEN1KMT2AALDH1A1MAPTXDH
SCHEMBL4259236 0.79 ALDH1A1 (0.50) CXCR1CXCR2ALDH1A1MAPTXDH
SCHEMBL3361866 0.79 LRRK2 (0.48) MEN1KMT2AALDH1A1MAPTGSK3B
SCHEMBL14393261 0.78 MEN1 (0.35) MEN1KMT2ATTRALBCXCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6300353-B1 FOR THERAPY OF FUNGAL INFECTIONS BASILEA PHARMACEUTICA AG, A SWISS COMPANY (CH) 2001-10-09 US disclosed
US-5958950-A CARDIOVASCULAR DISORDERS WARNER-LAMBERT COMPANY (US) 1999-09-28 US disclosed
WO-1999045008-A1 3-[4-(4-CYANOPHENYL)THIAZOL-2-Y)]-1-(1H-1,2,4-TRIAZOL-1-YL)-BUTAN-2-OL DERIVATIVES HAVING ANTIFUNGAL ACTIVITY F. HOFFMANN-LA ROCHE AG (CH) 1999-09-10 WO disclosed
WO-1997012615-A1 BENZIMIDAZOLE DERIVATIVES AS 15-LO INHIBITORS WARNER-LAMBERT COMPANY (US) 1997-04-10 WO disclosed