SCHEMBL7450868

SCHEMBL7450868

CCOC(=O)c1nc(C)n2c1CSc1cc(F)ccc1-2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 8/20 0.44
GABRB3 P28472 8/20 0.44
GABRA5 P31644 8/20 0.44
TSHR P16473 3/20 0.44
GABRA2 P47869 3/20 0.44
GABRB2 P47870 3/20 0.44
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 1/20 0.44
GABRP O00591 1/20 0.44
GABRD O14764 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
GABRA1 P14867 1/20 0.44
GABRB1 P18505 1/20 0.44
CYP2C19 P33261 1/20 0.44
GABRA3 P34903 1/20 0.44
GABRA4 P48169 1/20 0.44
GABRE P78334 1/20 0.44
KMT2A Q03164 1/20 0.44
GABRA6 Q16445 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7457553 0.87 GABRA2 (0.46) GABRG2GABRB3GABRA5GABRA2GABRB2
SCHEMBL7454157 0.85 HSD17B3 (0.44) ALDH1A1HSD17B3HTR7HPGDHSD17B10
SCHEMBL7452821 0.84 HSD17B3 (0.35) GABRG2GABRB3GABRA5TSHRGABRA2
SCHEMBL7454502 0.84 NPSR1 (0.48) GABRG2GABRB3GABRA5GABRA2ALDH1A1
SCHEMBL7449989 0.83 GLP1R (0.35) GABRG2GABRB3GABRA5TSHRGABRA2
SCHEMBL7458456 0.80 LMNA (0.45) GABRG2GABRB3GABRA5GABRA2GABRB2
SCHEMBL7453223 0.80 GABRG2 (0.45) GABRG2GABRB3GABRA5TSHRGABRA2
SCHEMBL7454183 0.79 GRM5 (0.40) GABRG2GABRB3GABRA5TSHRGABRA2
SCHEMBL7454766 0.78 GABRG2 (0.44) GABRG2GABRB3GABRA5TSHRGABRA2
SCHEMBL3604654 0.75 GLA (0.45) GABRG2GABRB3GABRA5TSHRGABRA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011151361-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-12-08 WO disclosed
WO-2011151361-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-12-08 WO disclosed