SCHEMBL7453085

SCHEMBL7453085

CCN(CC)C(=O)COc1ccc(-c2nsc3ccc(-n4c(=O)cc(C(F)(F)F)n(C)c4=O)cc23)cc1C

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 13/20 0.33
PPARA Q07869 7/20 0.33
PDE4B Q07343 1/20 0.33
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
AR P10275 1/20 0.32
ALDH1A1 P00352 2/20 0.32
PPARG P37231 4/20 0.32
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
MEN1 O00255 1/20 0.30
CYP3A4 P08684 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
ALOX15 P16050 1/20 0.30
KMT2A Q03164 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7459199 0.91 PPARD (0.33) PPARDPPARABCHEACHEPPARG
SCHEMBL7455505 0.90 OXTR (0.36) PPARDPPARAKDM4EMEN1MAPT
SCHEMBL7453077 0.88 TRPM8 (0.33) BCHEACHEALDH1A1KDM4EGAA
SCHEMBL7458904 0.84 PTGS2 (0.36) KDM4ETDP1MAPT
SCHEMBL7457864 0.84
SCHEMBL7461757 0.84
SCHEMBL7463328 0.84 KDM4E (0.31) ALDH1A1KDM4E
SCHEMBL7457226 0.82 HPGD (0.43) ALDH1A1KDM4ETDP1MEN1MAPT
SCHEMBL7453732 0.82 ALDH1A1 (0.33) ALDH1A1MAPTHPGD
SCHEMBL7462604 0.81 ESR1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0908457-B1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents BASF AG (DE) 2002-11-13 EP disclosed
EP-0908457-A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents American Cyanamid Company (US) 1999-04-14 EP disclosed