SCHEMBL7455378

SCHEMBL7455378

COC(=O)[C@H](Cc1ccc(O[Si](c2ccccc2)(c2ccccc2)C(C)(C)C)cc1)NCCNC(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 2/20 0.45
ITGB7 P26010 2/20 0.45
KLK5 Q9Y337 1/20 0.44
TDP1 Q9NUW8 2/20 0.42
PAX8 Q06710 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
CTSS P25774 4/20 0.42
CTSK P43235 3/20 0.42
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
MAPT P10636 2/20 0.40
POLB P06746 2/20 0.40
KDM4E B2RXH2 1/20 0.40
IDO1 P14902 1/20 0.40
MAPK1 P28482 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6936727 0.84 KLK5 (0.57) ITGA4ITGB7KLK5TDP1PAX8
SCHEMBL8497138 0.84 KLK5 (0.57) ITGA4ITGB7KLK5TDP1PAX8
SCHEMBL7452177 0.84 KLK5 (0.57) ITGA4ITGB7KLK5TDP1PAX8
SCHEMBL7455375 0.84 KLK5 (0.48) KLK5TDP1MEN1KMT2ACTSS
SCHEMBL5926274 0.83 CTSS (0.57) ITGA4ITGB7KLK5CTSSCTSK
SCHEMBL25832689 0.82 NAMPT (0.49) KMT2ACTSSCTSKMAPTIDO1
SCHEMBL27331529 0.78 CTSS (0.56) ITGA4ITGB7KLK5CTSSCTSK
SCHEMBL7520488 0.77 LTA4H (0.45) MEN1KMT2AHDAC8ALDH1A1LMNA
SCHEMBL30841324 0.77 ITGA4 (0.52) ITGA4ITGB7KLK5CTSSCTSK
SCHEMBL27332108 0.77 ITGA4 (0.52) ITGA4ITGB7KLK5CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973945-A4 CHIRAL PEPTIDE NUCLEIC ACIDS AND METHODS FOR PREPARING SAME ISIS PHARMACEUTICALS INC (US) 2002-07-17 EP disclosed
EP-0973945-A1 CHIRAL PEPTIDE NUCLEIC ACIDS AND METHODS FOR PREPARING SAME ISIS PHARMACEUTICALS, INC. (US) 2000-01-26 EP disclosed
US-6015887-A PREPARING SYNTHETIC MONOMERS BY DEHYDRATIVE COUPLING OF AMINE AND ALCOHOL STARTING REAGENTS ISIS PHARMACEUTICALS, INC. (US) 2000-01-18 US disclosed
WO-1998046794-A1 CHIRAL PEPTIDE NUCLEIC ACIDS AND METHODS FOR PREPARING SAME ISIS PHARMACEUTICALS, INC. (US) 1998-10-22 WO disclosed