SCHEMBL7459116

SCHEMBL7459116

COc1ccc(-c2nsc3ccc(-n4c(=O)cc(C)n(C)c4=O)cc23)cc1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD9 Q9H8M2 3/20 0.36
PTGS2 P35354 2/20 0.35
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
CYP19A1 P11511 3/20 0.32
NQO2 P16083 3/20 0.32
CYP2C9 P11712 1/20 0.32
MAP4K1 Q92918 1/20 0.31
PTGS1 P23219 1/20 0.31
STK17B O94768 1/20 0.31
USP2 O75604 1/20 0.30
TP53 P04637 1/20 0.30
TDP2 O95551 1/20 0.30
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30
SRC P12931 2/20 0.30
OXTR P30559 1/20 0.30
ABL1 P00519 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7458904 0.89 PTGS2 (0.36) BRD9PTGS2KDM4EMAPTCYP2C9
SCHEMBL7459099 0.84 BRD9 (0.36) BRD9MAPTCYP19A1NQO2CYP2C9
SCHEMBL7453460 0.81 TP53 (0.35) BRD9PTGS2MAPTCYP2C9PTGS1
SCHEMBL7460643 0.81 PTGS2 (0.35) BRD9PTGS2KDM4EMAPTCYP2C9
SCHEMBL7460298 0.81 TNF (0.37) BRD9PTGS2KDM4EMAPTCYP2C9
SCHEMBL7453732 0.79 ALDH1A1 (0.33) MAPT
SCHEMBL7455505 0.79 OXTR (0.36) KDM4EMAPTOXTR
SCHEMBL7462378 0.79 BCAT1 (0.44) PTGS2PTGS1
SCHEMBL7461247 0.78 PTGS1 (0.33) PTGS2KDM4EMAPTPTGS1TP53
SCHEMBL7457864 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0908457-B1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents BASF AG (DE) 2002-11-13 EP disclosed
EP-0908457-A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents American Cyanamid Company (US) 1999-04-14 EP disclosed
WO-1999014216-A1 SUBSTITUTED 3(-1,2-BENZISOTHIAZOL OR ISOXAZOL-5 YL)-SUBSTITUTED PYRIMIDINE AS HERBICIDES AMERICAN CYANAMID COMPANY (US) 1999-03-25 WO disclosed