SCHEMBL7460643

SCHEMBL7460643

COc1ccc(-c2nsc3ccc(-n4c(=O)cc(C(F)(F)F)n(C(C)C)c4=O)cc23)cc1C

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.35
PTGS1 P23219 1/20 0.35
SRC P12931 2/20 0.33
MAPT P10636 2/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
BRD9 Q9H8M2 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7458904 0.89 PTGS2 (0.36) PTGS2PTGS1MAPTLMNATP53
SCHEMBL7460631 0.86 GRM8 (0.31) CYP1A2CYP2C9BRD9
SCHEMBL7460298 0.86 TNF (0.37) PTGS2PTGS1MAPTLMNATP53
SCHEMBL7461247 0.83 PTGS1 (0.33) PTGS2PTGS1MAPTLMNATP53
SCHEMBL7453732 0.83 ALDH1A1 (0.33) MAPT
SCHEMBL7453460 0.81 TP53 (0.35) PTGS2PTGS1MAPTLMNATP53
SCHEMBL7459116 0.81 BRD9 (0.36) PTGS2PTGS1SRCMAPTTP53
SCHEMBL7462378 0.81 BCAT1 (0.44) PTGS2PTGS1
SCHEMBL7456944 0.79
SCHEMBL7455505 0.79 OXTR (0.36) MAPTCYP1A2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0908457-B1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents BASF AG (DE) 2002-11-13 EP disclosed
EP-0908457-A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents American Cyanamid Company (US) 1999-04-14 EP disclosed