SCHEMBL7459203

SCHEMBL7459203

CCOc1cccc(NC(=O)NS(=O)(=O)c2ccc(C)cc2)n1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.68
MAPK8 P45983 1/20 0.57
PKM P14618 1/20 0.56
KMT2A Q03164 2/20 0.53
ALDH1A1 P00352 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
LMNA P02545 3/20 0.52
NLRP3 Q96P20 1/20 0.52
MEN1 O00255 1/20 0.51
USP2 O75604 1/20 0.51
GAA P10253 1/20 0.48
PTGS1 P23219 1/20 0.48
PTGS2 P35354 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
FBP1 P09467 1/20 0.46
TP53 P04637 1/20 0.46
ALB P02768 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7459393 0.87 MAPK8 (0.53) KDM4EMAPK8PKMKMT2AALDH1A1
SCHEMBL6465388 0.81 KDM4E (1.00) KDM4EPKMKMT2AALDH1A1SMN1; SMN2
SCHEMBL7452165 0.81 LMNA (0.60) KDM4EPKMKMT2AALDH1A1SMN1; SMN2
SCHEMBL7455341 0.79 KDM4E (0.76) KDM4EPKMKMT2AALDH1A1SMN1; SMN2
SCHEMBL7458478 0.79 KDM4E (0.76) KDM4EPKMKMT2AALDH1A1SMN1; SMN2
SCHEMBL7460054 0.77 PKM (0.58) PKMKMT2AALDH1A1SMN1; SMN2LMNA
SCHEMBL8383136 0.74 HRH3 (0.65) KMT2AALDH1A1SMN1; SMN2LMNAMEN1
SCHEMBL24271910 0.74 MAPK8 (1.00) KDM4EMAPK8PKMKMT2ASMN1; SMN2
SCHEMBL10364805 0.73 KMT2A (0.58) KDM4EKMT2AALDH1A1SMN1; SMN2LMNA
SCHEMBL6463108 0.72 LMNA (0.64) KDM4EPKMKMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0819118-B1 POTASSIUM ION CHANNEL BLOCKERS POLYCHIP PHARMACEUTICALS PTY (AU) 2002-09-18 EP disclosed
US-5929082-A SULFONYL(THIO)UREA AND SULFONYLGUANIDINE COMPOUNDS; TREATMENT OF DIABETES, CARDIAC ARRHYTHMIAS, ISCHEMIA, HYPOXIC CARDIOVASCUALR DISORDERS AND CANCER POLYCHIP PHARMACEUTICALS PTY LTD (AU) 1999-07-27 US disclosed
EP-0819118-A4 POTASSIUM ION CHANNEL BLOCKERS POLYCHIP PHARMACEUTICALS PTY (AU) 1998-04-29 EP disclosed
EP-0819118-A1 POTASSIUM ION CHANNEL BLOCKERS Polychip Pharmaceuticals Pty. Ltd. (AU) 1998-01-21 EP disclosed
WO-1996030341-A1 POTASSIUM ION CHANNEL BLOCKERS POLYCHIP PHARMACEUTICALS PTY. LTD. (AU) 1996-10-03 WO disclosed