SCHEMBL7461966

SCHEMBL7461966

Cc1cc(-c2nsc3ccc(-n4c(=O)cc(C(F)(F)F)n(C)c4=O)cc23)ccc1OCCN1CCOCC1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.43
HTR2B P41595 4/20 0.43
HTR2A P28223 4/20 0.43
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
ADORA2A P29274 2/20 0.38
LSS P48449 2/20 0.37
OXTR P30559 1/20 0.37
AVPR1A P37288 1/20 0.37
MCHR1 Q99705 3/20 0.35
SYK P43405 1/20 0.35
P2RY12 Q9H244 1/20 0.35
PDE4B Q07343 1/20 0.35
HTR1A P08908 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7455505 0.86 OXTR (0.36) OXTRAVPR1A
SCHEMBL7458904 0.83 PTGS2 (0.36) MCHR1
SCHEMBL7463328 0.83 KDM4E (0.31)
SCHEMBL7457864 0.83
SCHEMBL7461757 0.83
SCHEMBL7453732 0.81 ALDH1A1 (0.33)
SCHEMBL7457226 0.80 HPGD (0.43) ADORA2A
SCHEMBL7459199 0.80 PPARD (0.33)
SCHEMBL7453085 0.80 PPARD (0.33) PDE4B
SCHEMBL7453460 0.79 TP53 (0.35) PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0908457-B1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents BASF AG (DE) 2002-11-13 EP disclosed
EP-0908457-A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents American Cyanamid Company (US) 1999-04-14 EP disclosed