SCHEMBL7463293

SCHEMBL7463293

CC(=O)C(C(N)=O)c1c(F)cccc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.39
KCNN4 O15554 5/20 0.37
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
CTSS P25774 2/20 0.36
CTSK P43235 1/20 0.36
NOTUM Q6P988 2/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
KIF11 P52732 1/20 0.35
PTGS2 P35354 1/20 0.35
CYP3A4 P08684 1/20 0.34
CD38 P28907 1/20 0.34
KCNH2 Q12809 1/20 0.34
KCNE1 P15382 1/20 0.34
KCNQ1 P51787 1/20 0.34
SLC9A1 P19634 1/20 0.33
EPHX2 P34913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7676477 0.88 AKR1C3 (0.41) KCNN4CES2CES1NOTUMAKR1C3
SCHEMBL7479581 0.85 CES2 (0.44) CES2CES1NOTUM
SCHEMBL7563011 0.81 CES2 (0.46) SCN9AKCNN4CES2CES1CTSS
SCHEMBL7470783 0.81 MAOB (0.37) CTSSCTSKNOTUMCYP3A4CD38
SCHEMBL7471669 0.76 ACP3 (0.44) KCNN4CTSSCTSKSLC9A1
SCHEMBL28722929 0.74 KCNN4 (0.34) SCN9AKCNN4CES2CES1CTSS
SCHEMBL14120994 0.73 P2RX7 (0.40) CTSSCTSKAKR1C3AKR1C2
SCHEMBL26620983 0.73 P2RX7 (0.40) CTSSCTSKAKR1C3AKR1C2
SCHEMBL7465798 0.72 CES2 (0.47) KCNN4CES2CES1AKR1C3AKR1C2
SCHEMBL7465792 0.72 CES2 (0.47) KCNN4CES2CES1AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077701-A4 ANTI-VIRAL COMPOUNDS LILLY CO ELI (US) 2002-03-20 EP disclosed
US-6358971-B1 FOR INHIBITING THE GROWTH OF A PICORNAVIRUS ELI LILLY AND COMPANY 2002-03-19 US disclosed
EP-1077701-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 2001-02-28 EP disclosed
WO-1999059587-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 1999-11-25 WO disclosed