SCHEMBL7465151

SCHEMBL7465151

CCCCC(c1ncccn1)c1cccc(F)c1F

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.34
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
PDE4D Q08499 1/20 0.32
TLR8 Q9NR97 4/20 0.31
F2RL1 P55085 3/20 0.31
CYP19A1 P11511 1/20 0.31
TSHR P16473 1/20 0.31
CTSA P10619 1/20 0.30
TLR7 Q9NYK1 1/20 0.30
GLS O94925 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19496643 0.74 CES2 (0.37) KCNH2CES2CES1TSHRGLS
SCHEMBL7786189 0.74 CES2 (0.44) KCNH2CES2CES1GLS
SCHEMBL16951255 0.73 CES2 (0.36) KCNH2CES2CES1GLSL3MBTL1
SCHEMBL15301598 0.73 CES2 (0.36) KCNH2CES2CES1GLSL3MBTL1
SCHEMBL8332508 0.73 SIGMAR1 (0.44) PDE4DCYP19A1TSHR
SCHEMBL11994152 0.72 CYP19A1 (0.43) CYP19A1L3MBTL1
SCHEMBL29206337 0.71 CES2 (0.39) CES2CES1GLS
SCHEMBL8746393 0.70 CES2 (0.42) CES2CES1GLS
SCHEMBL15107633 0.70 CES2 (0.33) KCNH2CES2CES1
SCHEMBL22932917 0.69 NR1I2 (0.38) CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0817773-B1 PYRIMIDINE COMPOUNDS QINETIQ LTD (GB) 2002-06-12 EP disclosed
US-6121448-A LIQUID CRYSTALLINE COMPOUNDS THE SECRETARY OF STATE FOR DEFENCE IN HER BRITTANIC MAJESTY'S GOVERNMENT OF THE UNITED KINGDOM OF GREAT BRITAIN AND NORTHERN IRELAND (GB) 2000-09-19 US disclosed
US-5986096-A REACTION OF HYDROGEN IODIDE WITH CHLORO-5-BROMOPYRIMIDINE THE SECRETARY OF STATE FOR DEFENCE IN HER BRITANNIC MAJESTY'S A GOVERNMENT OF THE U.K. OF GT. BRITAIN & N. IRELAND OF DEFENCE EVALUATION & RESEARCH AGENCY (GB) 1999-11-16 US disclosed
WO-1996030344-A2 PYRIMIDINE COMPOUNDS THE SECRETARY OF STATE FOR DEFENCE (GB) 1996-10-03 WO disclosed