SCHEMBL7470355

SCHEMBL7470355

COc1cccc(CCN2CCC(C3=CC(F)=CC[CH]3)CC2)c1OC

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.43
KCNH2 Q12809 3/20 0.43
HTR2A P28223 2/20 0.43
GRM2 Q14416 1/20 0.43
DRD2 P14416 1/20 0.43
ADRA2B P18089 1/20 0.43
DRD1 P21728 1/20 0.43
HTR2C P28335 1/20 0.43
HRH1 P35367 1/20 0.43
ADRA1B P35368 1/20 0.43
OPRK1 P41145 1/20 0.43
HTR2B P41595 1/20 0.43
KCNQ1 P51787 1/20 0.43
TMEM97 Q5BJF2 1/20 0.43
HRH3 Q9Y5N1 1/20 0.42
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
BACE1 P56817 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6603889 0.71 HTR2A (0.68) HTR2AGRM2DRD2DRD1HTR2C
SCHEMBL6603656 0.70 HTR2A (0.51) SIGMAR1KCNH2HTR2AGRM2DRD2
SCHEMBL8279384 0.69 HTR2A (0.62) KCNH2HTR2AGRM2DRD2ADRA2B
SCHEMBL3046365 0.65 HTR2B (0.74) SIGMAR1KCNH2HTR2ADRD2ADRA2B
SCHEMBL3046362 0.65 HTR2B (0.74) SIGMAR1KCNH2HTR2ADRD2ADRA2B
SCHEMBL5206867 0.65 HTR1A (0.83)
SCHEMBL17828187 0.65 SIGMAR1 (0.77) SIGMAR1KCNH2HRH3
SCHEMBL26807183 0.63 SIGMAR1 (0.52) SIGMAR1KCNH2DRD2HRH3
SCHEMBL16056564 0.63 KCNH2 (0.78) SIGMAR1KCNH2HRH3
SCHEMBL1991377 0.62 HTR2A (0.62) KCNH2HTR2AGRM2DRD2ADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1202966-A1 PIPERIDINE ALCOHOLS MERCK PATENT GmbH (DE) 2002-05-08 EP disclosed
WO-2001014332-A1 PIPERIDINE ALCOHOLS MERCK PATENT GMBH (DE) 2001-03-01 WO disclosed