SCHEMBL7472819

SCHEMBL7472819

CC(C)(C)OC(=O)Nc1ccccc1Cn1c(=O)n(S(=O)(=O)c2ccc(Cl)cc2)c(=O)c2ccc(Cl)cc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
HDAC6 Q9UBN7 3/20 0.38
PSEN1 P49768 2/20 0.38
PSEN2 P49810 2/20 0.38
APH1B Q8WW43 2/20 0.38
NCSTN Q92542 2/20 0.38
APH1A Q96BI3 2/20 0.38
PSENEN Q9NZ42 2/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC8 Q9BY41 2/20 0.38
RORC P51449 1/20 0.38
BRD4 O60885 1/20 0.37
CYP2C9 P11712 1/20 0.36
PTGER1 P34995 1/20 0.36
MAPK8 P45983 2/20 0.36
S1PR2 O95136 1/20 0.36
CMA1 P23946 1/20 0.36
NOD2 Q9HC29 1/20 0.35
NOD1 Q9Y239 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7467388 0.79 PSEN1 (0.42) HDAC6PSEN1PSEN2APH1BNCSTN
SCHEMBL7470720 0.78 PSEN1 (0.43) HDAC6PSEN1PSEN2APH1BNCSTN
SCHEMBL7457233 0.77 HDAC6 (0.39) HDAC6HDAC1HDAC8RORCMAPK8
SCHEMBL7457228 0.77 HDAC6 (0.39) HDAC6HDAC1HDAC8RORCMAPK8
SCHEMBL7469901 0.77 CMA1 (0.44) HDAC6PSEN1PSEN2APH1BNCSTN
Bromide SCHEMBL7465782 0.76 PSEN1 (0.37) HDAC6PSEN1PSEN2APH1BNCSTN
SCHEMBL7472667 0.76 TP53 (0.42) POLB
SCHEMBL7460713 0.76 MAPK8 (0.55) HDAC6PSEN1PSEN2APH1BNCSTN
SCHEMBL7472701 0.75 PSEN1 (0.42) HDAC6PSEN1PSEN2APH1BNCSTN
SCHEMBL7463851 0.75 NOX4 (0.46) MAPK8CMA1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795548-B1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LTD (JP) 2002-07-03 EP disclosed
US-5814631-A CHYMASE INHIBITOR, CARDIVASCULAR SUNTORY LIMITED (JP) 1998-09-29 US disclosed
EP-0795548-A1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LIMITED (JP) 1997-09-17 EP disclosed