SCHEMBL7473667

SCHEMBL7473667

COc1cccc2cc(C(=O)Nc3ccc4[nH]c(C(=O)N5C[C@@H](CCl)c6c5cc(O)c5[nH]c(C(F)(F)F)c(C(=O)O)c65)cc4c3)ncc12

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PYGL P06737 1/20 0.33
ABCB1 P08183 7/20 0.32
ABL1 P00519 1/20 0.32
SRC P12931 1/20 0.32
NR4A1 P22736 1/20 0.31
ENPP1 P22413 1/20 0.30
F11 P03951 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7461868 0.95 ABCB1 (0.32) PYGLABCB1ABL1SRCNR4A1
SCHEMBL7469597 0.90 PYGL (0.32) PYGLF11
SCHEMBL7473629 0.89 P4HB (0.34) ABCB1ENPP1F11
SCHEMBL7460763 0.89 KDM4E (0.37)
SCHEMBL7463553 0.89 KDM4E (0.36)
SCHEMBL7459606 0.88 ABL1 (0.32) PYGLABCB1ABL1SRC
SCHEMBL7475427 0.88 KMT2A (0.33) PYGLABCB1F11
SCHEMBL6627433 0.88 MAPT (0.38) PYGLABCB1
SCHEMBL7466678 0.86 GABRA1 (0.34)
SCHEMBL7458517 0.86 P4HB (0.34) ABCB1ENPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0656360-B1 TRIFLUOROMETHYLPYRROLOINDOLE CARBOXYLIC ESTER DERIVATIVE AND PROCESS FOR PRODUCING THE SAME KYORIN SEIYAKU KK (JP) 2002-11-20 EP disclosed
US-5629430-A ANTICARCINOGENIC AGENTS KYORIN PHARMACEUTICAL CO., LTD. (JP) 1997-05-13 US disclosed
EP-0656360-A1 TRIFLUOROMETHYLPYRROLOINDOLE CARBOXYLIC ESTER DERIVATIVE AND PROCESS FOR PRODUCING THE SAME KYORIN PHARMACEUTICAL CO., LTD. (JP) 1995-06-07 EP disclosed