SCHEMBL7474367

SCHEMBL7474367

CCOC(=O)c1ccccc1Cn1ccc2cc(OC(C)=O)ccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
TSHR P16473 1/20 0.43
BCL2 P10415 2/20 0.42
MCL1 Q07820 2/20 0.42
KDM4E B2RXH2 5/20 0.41
LMNA P02545 1/20 0.41
BRD4 O60885 1/20 0.41
ALDH1A1 P00352 4/20 0.41
HPGD P15428 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
FLT1 P17948 1/20 0.41
KDR P35968 1/20 0.41
GAA P10253 3/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
CDC25B P30305 1/20 0.40
GLA P06280 1/20 0.40
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7477071 0.86 THRA (0.52) BCL2MCL1KDM4EMEN1KMT2A
SCHEMBL7471302 0.85 TSHR (0.43) TSHRBCL2MCL1KDM4EALDH1A1
SCHEMBL7477507 0.85 CA12 (0.46) MAOAMAOBTSHRBCL2MCL1
SCHEMBL7481379 0.84 ALDH1A1 (0.46) TSHRKDM4EBRD4ALDH1A1HPGD
SCHEMBL27583585 0.84 LMNA (0.47) TSHRKDM4ELMNAALDH1A1HPGD
SCHEMBL7473999 0.83 PPARG (0.49) TSHRBCL2MCL1
SCHEMBL7478282 0.82 TSHR (0.42) TSHRKDM4ELMNAALDH1A1HPGD
SCHEMBL7474077 0.81 SERPINE1 (0.51) MAPT
SCHEMBL7483021 0.80 PPARD (0.58) MAOBBCL2MCL1MEN1KMT2A
SCHEMBL7482851 0.80 PPARG (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1379774-A Compounds ASTRAZENECA AB (SE) 2002-11-13 CN disclosed
EP-1210343-A2 BENZOIC ACID DERIVATIVES AND THEIR USE AS PPAR RECEPTOR AGONISTS AstraZeneca AB (SE) 2002-06-05 EP disclosed
WO-2001012187-A2 BENZOIC ACID DERIVATIVES AND THEIR USE AS PPAR RECEPTOR AGONISTS ASTRAZENECA AB (SE) 2001-02-22 WO disclosed
EP-0949921-A1 THROMBIN INHIBITORS Merck & Co., Inc. (US) 1999-10-20 EP disclosed
EP-0949921-A4 1999-10-20 EP disclosed
WO-1998006396-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 1998-02-19 WO disclosed