SCHEMBL7474672

SCHEMBL7474672

CC(=O)c1cc(C(F)(F)F)ccc1CC(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 6/20 0.51
RXRB P28702 3/20 0.51
RXRG P48443 3/20 0.51
NR1H2 P55055 3/20 0.46
NR1H3 Q13133 2/20 0.46
CES2 O00748 2/20 0.45
ALDH1A1 P00352 3/20 0.44
HPGD P15428 3/20 0.44
HSD17B10 Q99714 3/20 0.44
KDM4E B2RXH2 2/20 0.44
USP2 O75604 1/20 0.44
CYP2C19 P33261 1/20 0.44
POLQ O75417 2/20 0.44
PSEN1 P49768 1/20 0.43
PSEN2 P49810 1/20 0.43
APH1B Q8WW43 1/20 0.43
NCSTN Q92542 1/20 0.43
APH1A Q96BI3 1/20 0.43
PSENEN Q9NZ42 1/20 0.43
AGBL2 Q5U5Z8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2337724 0.87 ALDH1A1 (0.53) RXRARXRBRXRGNR1H2NR1H3
SCHEMBL7472612 0.86 CES2 (0.44) RXRARXRBRXRGNR1H2NR1H3
SCHEMBL8916995 0.83 CFTR (0.46) RXRANR1H2NR1H3CES2ALDH1A1
SCHEMBL17899450 0.81 RXRA (0.72) RXRARXRBRXRGNR1H2NR1H3
SCHEMBL3135089 0.80 RXRA (0.53) RXRARXRBRXRGCES2ALDH1A1
SCHEMBL3741058 0.78 POLQ (0.61) RXRARXRBRXRGCES2POLQ
SCHEMBL30716953 0.78 POLQ (0.61) RXRARXRBRXRGCES2POLQ
SCHEMBL30530542 0.78 IDO1 (0.51) RXRARXRBRXRGALDH1A1HPGD
SCHEMBL512428 0.78 IDO1 (0.51) RXRARXRBRXRGALDH1A1HPGD
SCHEMBL27905706 0.78 RXRA (0.51) RXRARXRBRXRGNR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077701-A4 ANTI-VIRAL COMPOUNDS LILLY CO ELI (US) 2002-03-20 EP disclosed
EP-1077701-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 2001-02-28 EP disclosed
WO-1999059587-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 1999-11-25 WO disclosed