SCHEMBL7475083

SCHEMBL7475083

COC(=O)c1cc(-c2ccc(Cl)cc2F)nn1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA9 Q16790 1/20 0.48
KMO O15229 2/20 0.43
ALPL P05186 2/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
GRIN2B Q13224 1/20 0.40
ALDH1A1 P00352 2/20 0.39
DPP4 P27487 1/20 0.39
KDM4E B2RXH2 2/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
HSD17B10 Q99714 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11073103 0.80 CYP1A2 (0.53) CA12CA1CA2CA9CYP1A2
SCHEMBL6319050 0.76 KMO (0.43) KMOGRIN2B
SCHEMBL8165871 0.76 CA12 (0.41) CA12CA1CA2CA9KMO
SCHEMBL10960418 0.76 CA12 (0.47) CA12CA1CA2CA9CYP1A2
SCHEMBL7707702 0.76 KMO (0.42) KMOGRIN2B
SCHEMBL7474145 0.76 ALDH1A1 (0.40) KMOALPLALDH1A1DPP4KDM4E
SCHEMBL30722849 0.74 HDAC3 (0.56) CA12CA1CA2CA9ALDH1A1
SCHEMBL9081963 0.74 KMO (0.40) KMOGRIN2B
SCHEMBL28906210 0.73 ALDH1A1 (0.48) ALPLALDH1A1KDM4EGAAHPGD
SCHEMBL14800515 0.73 MAPT (0.50) ALPLCYP1A2CYP2C19DPP4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0769008-B1 PYRAZOLE DERIVATIVES AS HERBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2002-05-22 EP disclosed
US-6083881-A Pyrazole derivatives as herbicides NOVARTIS CORPORATION (US) 2000-07-04 US disclosed
EP-0769008-A1 PYRAZOLE DERIVATIVES AS HERBICIDES Novartis AG (CH) 1997-04-23 EP disclosed
WO-1996001254-A1 PYRAZOLE DERIVATIVES AS HERBICIDES CIBA-GEIGY AG (CH) 1996-01-18 WO disclosed