SCHEMBL7475210

SCHEMBL7475210

Nc1cccc2[nH]c(CCN3C(=O)c4ccccc4C3=O)nc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 4/20 0.48
CHEK1 O14757 1/20 0.45
ALDH1A1 P00352 3/20 0.45
MAPT P10636 6/20 0.44
GAA P10253 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
PKM P14618 1/20 0.40
TDP1 Q9NUW8 2/20 0.40
POLB P06746 2/20 0.40
CASP3 P42574 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7955816 0.87 CHEK1 (0.47) CHEK1ALDH1A1MAPTGAAMEN1
SCHEMBL7479144 0.81 GAA (0.46) PDE10AALDH1A1MAPTGAAMEN1
SCHEMBL5864478 0.80 ALDH1A1 (0.64) PDE10AALDH1A1MAPTGAAMEN1
SCHEMBL7964155 0.73 CHEK1 (0.58) PDE10ACHEK1MAPTGAAMEN1
SCHEMBL7481575 0.73 HTR6 (0.47) CHEK1MAPTGAAMEN1KMT2A
SCHEMBL6994637 0.72 CHEK1 (0.56) CHEK1ALDH1A1MAPTGAAMEN1
SCHEMBL12202119 0.72 ALDH1A1 (0.68) PDE10AALDH1A1MAPTRAB9ANPC1
SCHEMBL5736933 0.71 CHEK1 (0.55) PDE10ACHEK1ALDH1A1MAPTGAA
SCHEMBL7967546 0.70 CHEK1 (0.51) PDE10ACHEK1MAPTGAAMEN1
SCHEMBL3938941 0.70 CHEK1 (0.57) PDE10ACHEK1ALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207693-B1 Benzamide derivatives having a vasopressin antagonistic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-03-27 US disclosed
EP-0946519-A1 BENZAMIDE DERIVATIVES HAVING A VASOPRESSIN ANTAGONISTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-06 EP disclosed
WO-1998024771-A1 BENZAMIDE DERIVATIVES HAVING A VASOPRESSIN ANTAGONISTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-06-11 WO disclosed