SCHEMBL7476772

SCHEMBL7476772

O=C(O)N(c1ccc2c(c1F)CN(Nc1ccncc1)C2)N1CCc2ccccc2C1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 1/20 0.34
LIPE Q05469 1/20 0.33
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
EED O75530 1/20 0.33
NAMPT P43490 2/20 0.33
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
PRMT5 O14744 2/20 0.32
WDR77 Q9BQA1 2/20 0.32
SLC22A12 Q96S37 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7485803 0.89 LIPE (0.35) TRPM8LIPENPC1RAB9ATP53
Hydrochloric Acid SCHEMBL7484862 0.88 LIPE (0.35) TRPM8LIPENPC1RAB9ATP53
SCHEMBL7482587 0.82 GRIN2D (0.37) TRPM8LIPENPC1RAB9ATP53
Hydrochloric Acid SCHEMBL7479742 0.74 LIPE (0.51) TRPM8LIPENPC1RAB9AEED
SCHEMBL7477612 0.72 NAMPT (0.42) SMN1; SMN2NAMPTHPGDCYP1A2CYP3A4
SCHEMBL7477903 0.70 EED (0.54) LIPENPC1RAB9ATP53SMN1; SMN2
SCHEMBL7534680 0.69 NAMPT (0.33) SMN1; SMN2NAMPTGAAKDM4EALDH1A1
SCHEMBL7477144 0.69 NISCH (0.31) KMT2A
Bromide SCHEMBL7480922 0.68 NISCH (0.30)
SCHEMBL7481285 0.68 SLC6A2 (0.47) EEDNAMPTGRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950056-B1 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP claimed