SCHEMBL7476799

SCHEMBL7476799

COc1ccc2c(c1)C(=O)N(Nc1ccncc1)C(=O)C2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
HPGD P15428 3/20 0.51
GAA P10253 2/20 0.51
KDM4E B2RXH2 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
KMT2A Q03164 3/20 0.50
MEN1 O00255 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
CASP1 P29466 1/20 0.48
CASP6 P55212 1/20 0.48
CYP19A1 P11511 8/20 0.44
METAP1 P53582 2/20 0.43
CYP11B2 P19099 2/20 0.41
ADAM17 P78536 2/20 0.40
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8418434 0.98 ALDH1A1 (0.49) ALDH1A1HPGDGAAKDM4ECYP1A2
Hydrochloric Acid SCHEMBL8418433 0.98 ALDH1A1 (0.49) ALDH1A1HPGDGAAKDM4ECYP1A2
Hydrochloric Acid SCHEMBL7482266 0.96 ALDH1A1 (0.48) ALDH1A1HPGDGAAKDM4ECYP1A2
SCHEMBL7487924 0.84 CASP6 (0.51) ALDH1A1HPGDGAACYP1A2KMT2A
SCHEMBL8860233 0.82 CYP19A1 (0.43) ALDH1A1HPGDKMT2AMEN1SMN1; SMN2
SCHEMBL7479666 0.82 APP (0.46) ALDH1A1CYP1A2SMN1; SMN2CYP19A1LMNA
SCHEMBL7486935 0.81 CASP6 (0.51) KDM4ECYP1A2CASP6CYP19A1LMNA
SCHEMBL7479829 0.81 CASP6 (0.51) KDM4EKMT2AMEN1CASP6LMNA
Hydrochloric Acid SCHEMBL7485356 0.81 APP (0.45) ALDH1A1CYP1A2SMN1; SMN2CYP19A1LMNA
SCHEMBL7487129 0.78 ALDH1A1 (0.55) ALDH1A1HPGDGAAKDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0950056-A2 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS HOECHST MARION ROUSSEL, INC. (US) 1999-10-20 EP claimed
WO-1998029407-A2 N-(PYRIDINYLAMINO)ISOINDOLINES FOR TREATING ALZHEIMER'S AND DEPRESSION HOECHST MARION ROUSSEL, INC. (US) 1998-07-09 WO claimed
EP-0950056-B1 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP disclosed
EP-0950056-A2 N-(PYRIDINYLAMINO)ISOINDOLINES AND RELATED COMPOUNDS HOECHST MARION ROUSSEL, INC. (US) 1999-10-20 EP disclosed
WO-1998029407-A2 N-(PYRIDINYLAMINO)ISOINDOLINES FOR TREATING ALZHEIMER'S AND DEPRESSION HOECHST MARION ROUSSEL, INC. (US) 1998-07-09 WO disclosed