SCHEMBL7478153

SCHEMBL7478153

CCC(c1cc(OC)c(OC)c(OC)c1)C(CC(N)=O)C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.43
MAPK1 P28482 1/20 0.43
PDE4A P27815 2/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
TNF P01375 1/20 0.39
MAPT P10636 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38
PTGS2 P35354 1/20 0.38
POLB P06746 1/20 0.38
TSHR P16473 1/20 0.37
APOBEC3A P31941 1/20 0.37
HTT P42858 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
PDK1 Q15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29276367 0.79 L3MBTL1 (0.43) L3MBTL1MAPK1PDE4APDE4BPDE4C
SCHEMBL11437458 0.72 ALDH1A1 (0.50) L3MBTL1MAPK1MAPTKDM4EMEN1
SCHEMBL2930054 0.72 MAPT (0.49) L3MBTL1MAPK1MAPTKDM4EALDH1A1
SCHEMBL18925030 0.71 PTGS2 (0.50) L3MBTL1MAPK1MAPTPTGS2
SCHEMBL7290682 0.70 PDK1 (0.46) L3MBTL1MAPK1MAPTKDM4EALDH1A1
SCHEMBL7427374 0.69 CES2 (0.42)
SCHEMBL2924476 0.68 POLB (0.50) L3MBTL1MAPK1MAPTKDM4EMEN1
SCHEMBL7354148 0.68 CA12 (0.45) MEN1KMT2A
SCHEMBL24983762 0.67 L3MBTL1 (0.50) L3MBTL1MAPK1MAPTKDM4EMEN1
SCHEMBL500044 0.67 AKR1C3 (0.54) L3MBTL1MAPK1MAPTKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082127-A4 SUCCINAMIDE INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME WARNER LAMBERT CO (US) 2002-10-09 EP claimed
EP-1082127-A1 SUCCINAMIDE INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME WARNER-LAMBERT COMPANY (US) 2001-03-14 EP claimed
WO-1999056765-A1 SUCCINAMIDE INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME WARNER-LAMBERT COMPANY (US) 1999-11-11 WO claimed