SCHEMBL7480428

SCHEMBL7480428

CCCCCN1CC=C(c2c[nH]c3ccc(NC(=O)COc4ccccc4)cc23)CC1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.51
HTR1A P08908 6/20 0.51
HTR2A P28223 2/20 0.51
NOS3 P29474 2/20 0.51
NOS1 P29475 2/20 0.51
MAPT P10636 1/20 0.50
SLC6A4 P31645 3/20 0.49
HTR7 P34969 3/20 0.49
HTR6 P50406 3/20 0.49
DRD4 P21917 1/20 0.49
HTR2C P28335 1/20 0.49
DRD3 P35462 1/20 0.49
HTR2B P41595 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7483579 0.92 DRD2 (0.49) DRD2HTR1AHTR2ANOS3NOS1
SCHEMBL7485964 0.88 DRD2 (0.47) DRD2HTR1AHTR2ANOS3NOS1
SCHEMBL7487821 0.87 DRD2 (0.51) DRD2HTR1AHTR2ANOS3NOS1
SCHEMBL7477774 0.87 NOS3 (0.52) DRD2HTR1AHTR2ANOS3NOS1
SCHEMBL7477377 0.86 NOS3 (0.63) DRD2HTR1AHTR2ANOS3NOS1
SCHEMBL7480321 0.86 SIGMAR1 (0.52) DRD2HTR1AHTR2ANOS3NOS1
SCHEMBL7482362 0.85 NOS3 (0.62) DRD2HTR1AHTR2ANOS3NOS1
Glycolic Acid SCHEMBL30908796 0.85 NOS3 (0.51) DRD2HTR1AHTR2ANOS3NOS1
SCHEMBL7480418 0.85 MAPT (0.52) DRD2HTR1AHTR2ANOS3NOS1
SCHEMBL7476819 0.84 MAPT (0.48) DRD2HTR1AHTR2AMAPTSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260125645-A1 METHODS AND PHARMACOLOGICAL AGENTS FOR INCREASING EXPANSION, ENGRAFTMENT OR IMMUNE OUTPUT OF HUMAN HEMATOPOIETIC STEM CELLS IN TRANSPLANTATION AND DISEASE SETTINGS VALORISATION HSJ LP (CA) 2026-05-07 US disclosed
EP-0733628-B9 5-Substituted-3-(1,2,3,6-tetrahydropyridin-4-yl)- and 3-(piperidin-4-yl)-1H-indoles: 5-HT1F agonists LILLY CO ELI (US) 2002-06-12 EP disclosed
EP-0733628-B1 5-Substituted-3-(1,2,3,6-tetrahydropyridin-4-yl)- and 3-(piperidin-4-yl)-1H-indoles: 5-HT1F agonists LILLY CO ELI (US) 2000-12-27 EP disclosed
US-5962474-A ANALGESICS; HEADACHES ELI LILLY AND COMPANY (US) 1999-10-05 US disclosed
US-5708008-A TREATMENT OF MIGRAINE ELI LILLY AND COMPANY (US) 1998-01-13 US disclosed
WO-1996029075-A1 5-SUBSTITUTED-3-(1,2,3,6-TETRAHYDROPYRIDIN-4-YL)- AND 3-(PIPERIDIN-4-YL)-1H-INDOLES: NEW 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 1996-09-26 WO disclosed
EP-0733628-A1 5-Substituted-3-(1,2,3,6-tetrahydropyridin-4-yl)- and 3-(piperidin-4-yl)-1h-indoles: new 5-ht1f agonists ELI LILLY AND COMPANY (US) 1996-09-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260125645-A1 METHODS AND PHARMACOLOGICAL AGENTS FOR INCREASING EXPANSION, ENGRAFTMENT OR IMMUNE OUTPUT OF HUMAN HEMATOPOIETIC STEM CELLS IN TRANSPLANTATION AND DISEASE SETTINGS HTR1F, HTR1A, HTR1D DRD2 691/4885HTR1A 2/4885HTR2A 12/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.