SCHEMBL7482907

SCHEMBL7482907

Cc1nc(-c2ccc(N3CC(CN4CCN(S(=O)(=O)c5ccccc5C#N)CC4)OC3=O)cc2)no1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.44
GBA1 P04062 2/20 0.43
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 1/20 0.40
SIGMAR1 Q99720 5/20 0.40
PKM P14618 1/20 0.39
P2RX3 P56373 1/20 0.38
HTT P42858 1/20 0.37
KDM2B Q8NHM5 1/20 0.37
CTDSP1 Q9GZU7 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37
MAPT P10636 1/20 0.37
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7386638 0.89 THRB (0.47) THRBSIGMAR1P2RX3MAPT
SCHEMBL7388878 0.87 MAPT (0.46) THRBALDH1A1SIGMAR1P2RX3MAPT
SCHEMBL7392425 0.86 THRB (0.44) THRBGBA1ALDH1A1SIGMAR1P2RX3
SCHEMBL7388548 0.85 MAPT (0.45) THRBGBA1ALDH1A1SIGMAR1P2RX3
SCHEMBL7380624 0.85 PKM (0.44) THRBGBA1KDM4EALDH1A1SIGMAR1
SCHEMBL7387950 0.84 THRB (0.45) THRBSIGMAR1P2RX3HTTTSHR
SCHEMBL7390212 0.84 P2RX3 (0.43) THRBSIGMAR1P2RX3KDM2BMAPT
SCHEMBL7389109 0.84 THRB (0.51) THRBSIGMAR1MAPT
SCHEMBL7389428 0.84 THRB (0.45) THRBSIGMAR1P2RX3MAPT
SCHEMBL7381271 0.83 SIGMAR1 (0.46) THRBSIGMAR1HTTGAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056743-A1 BENZAMINE DERIVATIVES MERCK PATENT GmbH (DE) 2000-12-06 EP disclosed
WO-1999031092-A1 BENZAMINE DERIVATIVES MERCK PATENT GMBH (DE) 1999-06-24 WO disclosed