SCHEMBL7486143

SCHEMBL7486143

CC1(C)CCC(=O)c2c(-c3ccncc3)n[nH]c21

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 9/20 0.39
ALPL P05186 4/20 0.39
CDC7 O00311 1/20 0.36
CCNE2 O96020 1/20 0.36
CDK4 P11802 1/20 0.36
CCND1 P24385 1/20 0.36
CCNE1 P24864 1/20 0.36
CDK2 P24941 1/20 0.36
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
MAPK11 Q15759 3/20 0.35
MAPK14 Q16539 3/20 0.35
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480513 0.87 ATM (0.41) ALPLPDE3BPDE3ANPC1
SCHEMBL7484888 0.78 ROCK2 (0.42) LRRK2ALPLCDC7CCNE2CDK4
SCHEMBL7485161 0.77 CYP17A1 (0.34) LRRK2ALPL
SCHEMBL7484067 0.76 GAA (0.50) ALPL
SCHEMBL7482943 0.75 HSP90AA1 (0.39) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL7486190 0.75 POLL (0.39) ALPL
SCHEMBL7487084 0.75 HTR7 (0.41) ALPLNPC1
SCHEMBL7685046 0.74 CDC7 (0.51) CDC7
SCHEMBL7479968 0.70 ALPL (0.73) ALPL
SCHEMBL7485922 0.67 PARP1 (0.50) ALPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed