SCHEMBL7486332

SCHEMBL7486332

CN(CCC#N)S(=O)(=O)c1ccc2c(c1)C(=O)C(=O)N2

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 9/20 0.68
MAOA P21397 3/20 0.59
MAOB P27338 2/20 0.59
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA9 Q16790 1/20 0.49
ALDH1A1 P00352 2/20 0.45
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
CASP9 P55211 1/20 0.44
GAA P10253 1/20 0.43
KMT2A Q03164 3/20 0.43
RXFP1 Q9HBX9 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
TGM2 P21980 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7566978 0.84 CASP3 (0.74) CASP3MAOAMAOBCA12CA1
SCHEMBL6535335 0.81 CASP3 (1.00) CASP3MAOAMAOBCA12CA1
SCHEMBL6535436 0.79 CASP3 (0.67) CASP3MAOAMAOBCA12CA1
SCHEMBL6946269 0.78 PKLR (0.44) CASP3MAOAMAOBALDH1A1GAA
SCHEMBL4411083 0.78 CASP3 (0.64) CASP3MAOAMAOBCA12CA1
SCHEMBL7736087 0.77 CASP3 (0.64) CASP3MAOAMAOBCA12CA1
SCHEMBL4906814 0.76 MAOA (0.78) CASP3MAOAMAOBCA12CA1
SCHEMBL8312045 0.73 CASP3 (0.59) CASP3MAOAMAOBCA12CA1
SCHEMBL7204403 0.71 PDE4D (0.60) ALDH1A1KMT2A
SCHEMBL7601554 0.71 CASP3 (0.58) CASP3MAOAMAOBCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403792-B1 INHIBIT PRODUCTION OF CASPASE 3 AND 7 IN MAMMALS SMITHKLINE BEECHAM CORPORATION 2002-06-11 US claimed
EP-1001933-A4 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORP (US) 2002-11-06 EP disclosed
US-6403792-B1 INHIBIT PRODUCTION OF CASPASE 3 AND 7 IN MAMMALS SMITHKLINE BEECHAM CORPORATION 2002-06-11 US disclosed
EP-1001933-A1 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999006367-A1 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORPORATION (US) 1999-02-11 WO disclosed