SCHEMBL7736087

SCHEMBL7736087

CN(CCc1ccncc1)S(=O)(=O)c1ccc2c(c1)C(=O)C(=O)N2

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 9/20 0.64
MAOA P21397 5/20 0.58
MAOB P27338 4/20 0.58
PDE3B Q13370 2/20 0.50
PDE3A Q14432 2/20 0.50
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
NAMPT P43490 1/20 0.43
CASP7 P55210 2/20 0.42
TGM2 P21980 1/20 0.42
CASP1 P29466 1/20 0.41
CASP9 P55211 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6535436 0.88 CASP3 (0.67) CASP3MAOAMAOBCA12CA1
SCHEMBL7566978 0.81 CASP3 (0.74) CASP3MAOAMAOBCA12CA1
SCHEMBL6949029 0.80 PKLR (0.42) CASP3MAOAMAOBNAMPTGAA
SCHEMBL6535335 0.78 CASP3 (1.00) CASP3MAOAMAOBCA12CA1
SCHEMBL7486332 0.77 CASP3 (0.68) CASP3MAOAMAOBCA12CA1
SCHEMBL4906814 0.76 MAOA (0.78) CASP3MAOAMAOBCA12CA1
SCHEMBL4411083 0.75 CASP3 (0.64) CASP3MAOAMAOBCA12CA1
SCHEMBL14111824 0.73 SMN1; SMN2 (0.57) PDE3BPDE3ACA12CA1CA2
SCHEMBL2333739 0.73 TDP1 (0.60) CA12CA1CA2CA9NAMPT
SCHEMBL11174132 0.73 TDP1 (0.51) NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403792-B1 INHIBIT PRODUCTION OF CASPASE 3 AND 7 IN MAMMALS SMITHKLINE BEECHAM CORPORATION 2002-06-11 US claimed
US-6403792-B1 INHIBIT PRODUCTION OF CASPASE 3 AND 7 IN MAMMALS SMITHKLINE BEECHAM CORPORATION 2002-06-11 US disclosed