SCHEMBL7486567

SCHEMBL7486567

CSc1ccc(-c2ccccc2C(=O)C(=O)c2ccccc2)cc1F

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.42
ALOX5AP P20292 5/20 0.39
FEN1 P39748 5/20 0.39
ACMSD Q8TDX5 1/20 0.39
CES2 O00748 3/20 0.37
CES1 P23141 3/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
STK17B O94768 1/20 0.36
LTB4R2 Q9NPC1 1/20 0.36
TP53 P04637 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HTT P42858 1/20 0.35
SLC6A2 P23975 1/20 0.35
MAPT P10636 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28987613 0.77 ERN1 (0.41) ALOX5APFEN1ACMSDCES2CES1
SCHEMBL7089420 0.77 SLC6A4 (0.39) ARCES2CES1SLC6A4SLC6A3
SCHEMBL7085294 0.75 SLC6A4 (0.37) ARCES2CES1SLC6A4SLC6A3
Benzene SCHEMBL28343003 0.73 BCAT2 (0.55) CES2CES1SLC6A3MAPTALDH1A1
Biphenyl SCHEMBL28340553 0.73 BCAT2 (0.55) CES2CES1SLC6A3MAPTALDH1A1
SCHEMBL27676197 0.73 BCAT2 (0.59) CES2CES1HTTALDH1A1
SCHEMBL30277841 0.73 BCAT2 (0.59) CES2CES1HTTALDH1A1
SCHEMBL7085149 0.73 PTGS2 (0.40)
SCHEMBL981885 0.72 CES2 (0.63) CES2CES1LTB4R2MAPT
Water SCHEMBL6671736 0.72 SLC6A2 (0.57) ACMSDCES2CES1SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1211244-A2 4,5-substitued imidazolyl compounds for the treatment of inflammation G.D. Searle & Co. (US) 2002-06-05 EP disclosed