SCHEMBL7488160

SCHEMBL7488160

CC(C)(C)OC(=O)n1cnc(C[C@H](N)C(=O)O)c1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.42
CPB2 Q96IY4 14/20 0.41
CPB1 P15086 8/20 0.41
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30786466 0.87 CPB2 (0.37) CPB2CPB1
SCHEMBL18346836 0.86 CPB2 (0.42) CPB2CPB1
SCHEMBL25469012 0.86 CPB2 (0.42) CPB2CPB1
SCHEMBL20759177 0.85 CPB2 (0.39) CPB2CPB1
SCHEMBL30643159 0.84 CPB2 (0.36) CPB2CPB1
SCHEMBL10659919 0.83 CPB2 (0.46) CPB2CPB1
SCHEMBL3008885 0.81 ITGB3 (0.45) CPB2CPB1
SCHEMBL3008889 0.81 ITGB3 (0.45) CPB2CPB1
SCHEMBL13650201 0.81 ITGB3 (0.45) CPB2CPB1
SCHEMBL7001068 0.81 SLC7A5 (0.44) SLC7A5CPB2CPB1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3916000-B1 METHOD FOR PRODUCING PEPTIDE COMPOUND, PROTECTING GROUP-FORMING REAGENT, AND AROMATIC HETEROCYCLIC COMPOUND FUJIFILM CORP (JP) 2026-04-08 EP disclosed
US-20260034237-A1 LINKERS, DRUG LINKERS AND CONJUGATES THEREOF AND METHODS OF USING THE SAME GENMAB AS (DK) 2026-02-05 US disclosed
EP-4598592-A1 A COMPOUND AND ITS USE FOR DETECTING A DISEASE IN THE EXHALED BREATH OF A SUBJECT Owlstone Medical Limited (GB) 2025-08-13 EP disclosed
US-12325727-B2 Method for producing peptide compound, protective group-forming reagent, and aromatic heterocyclic compound FUJIFILM CORPORATION (JP) 2025-06-10 US disclosed
US-12227542-B2 Method for producing peptide compound, protective group-forming reagent, and condensed polycyclic compound FUJIFILM CORPORATION (JP) 2025-02-18 US disclosed
US-20240325561-A1 PEGYLATED DRUG-LINKERS FOR IMPROVED LIGAND-DRUG CONJUGATE PHARMACOKINETICS SEAGEN INC (US) 2024-10-03 US disclosed
US-20240261427-A1 LINKERS, DRUG LINKERS AND CONJUGATES THEREOF AND METHODS OF USING THE SAME PROFOUNDBIO US CO. 2024-08-08 US disclosed
US-20240245796-A1 LINKERS, DRUG LINKERS AND CONJUGATES THEREOF AND METHODS OF USING THE SAME PROFOUNDBIO US CO. 2024-07-25 US disclosed
US-20240207429-A1 LINKERS, DRUG LINKERS AND CONJUGATES THEREOF AND METHODS OF USING THE SAME WILMINGTON TRUST, NATIONAL ASSOCIATION 2024-06-27 US disclosed
US-20240207418-A1 LINKERS, DRUG LINKERS AND CONJUGATES THEREOF AND METHODS OF USING THE SAME PROFOUNDBIO US CO. 2024-06-27 US disclosed
EP-4269422-A1 METHOD FOR PRODUCING PEPTIDE COMPOUND CONTAINING N-SUBSTITUTED-AMINO ACID RESIDUE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2023-11-01 EP disclosed
CN-112010961-B Solid-liquid synthesis method of somalupeptide 深圳市健元医药科技有限公司 2023-05-16 CN disclosed
WO-2023068296-A1 METHOD FOR PRODUCING COMPOUNDS, METHOD FOR PRODUCING COMPOUND LIBRARY, COMPOUND LIBRARY, AND SCREENING METHOD 国立大学法人東京大学 2023-04-27 WO disclosed
WO-2022138891-A1 METHOD FOR PRODUCING PEPTIDE COMPOUND CONTAINING N-SUBSTITUTED-AMINO ACID RESIDUE 中外製薬株式会社 2022-06-30 WO disclosed
EP-3992187-A1 METHOD FOR PRODUCING PEPTIDE COMPOUND, REAGENT FOR FORMING PROTECTIVE GROUP, AND FUSED POLYCYCLIC COMPOUND FUJIFILM Corporation (JP) 2022-05-04 EP disclosed
US-20220112234-A1 METHOD FOR PRODUCING PEPTIDE COMPOUND, PROTECTIVE GROUP-FORMING REAGENT, AND CONDENSED POLYCYCLIC COMPOUND FUJIFILM CORPORATION (JP) 2022-04-14 US disclosed
US-20220072146-A1 PEGYLATED DRUG-LINKERS FOR IMPROVED LIGAND-DRUG CONJUGATE PHARMACOKINETICS SEAGEN INC (US) 2022-03-10 US disclosed
WO-2019139028-A1 RESIN COMPOSITION FOR INSULATING FILM 日産化学株式会社 2019-07-18 WO disclosed
EP-1242420-A2 AGENTS AND METHODS FOR THE TREATMENT OF PROLIFERATIVE DISEASES ELI LILLY AND COMPANY (US) 2002-09-25 EP disclosed
WO-2001044247-A2 AGENTS AND METHODS FOR THE TREATMENT OF PROLIFERATIVE DISEASES ELI LILLY AND COMPANY (US) 2001-06-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12227542-B2 Method for producing peptide compound, protective group-forming reagent, and condensed polycyclic compound C9, GRPR, VIP SLC7A5 2929/4885CPB2 803/4885CPB1 1295/4885
US-20260034237-A1 LINKERS, DRUG LINKERS AND CONJUGATES THEREOF AND METHODS OF USING THE SAME CSGALNACT1, SLC43A1, OSTC SLC7A5 54/4885CPB2 2596/4885CPB1 2091/4885
US-20240207418-A1 LINKERS, DRUG LINKERS AND CONJUGATES THEREOF AND METHODS OF USING THE SAME PAICS, DHFR, CD44 SLC7A5 378/4885CPB2 2555/4885CPB1 2381/4885
US-20220072146-A1 PEGYLATED DRUG-LINKERS FOR IMPROVED LIGAND-DRUG CONJUGATE PHARMACOKINETICS EGFR, HDGF, CD47 SLC7A5 318/4885CPB2 3396/4885CPB1 3113/4885
US-12325727-B2 Method for producing peptide compound, protective group-forming reagent, and aromatic heterocyclic compound HM13, MCHR1, QRFPR SLC7A5 2326/4885CPB2 1191/4885CPB1 713/4885
US-20240207429-A1 LINKERS, DRUG LINKERS AND CONJUGATES THEREOF AND METHODS OF USING THE SAME PAICS, DHFR, CD44 SLC7A5 378/4885CPB2 2555/4885CPB1 2381/4885
US-20240325561-A1 PEGYLATED DRUG-LINKERS FOR IMPROVED LIGAND-DRUG CONJUGATE PHARMACOKINETICS EGFR, HDGF, CD47 SLC7A5 316/4885CPB2 3379/4885CPB1 3105/4885
US-20240261427-A1 LINKERS, DRUG LINKERS AND CONJUGATES THEREOF AND METHODS OF USING THE SAME PAICS, DHFR, CD44 SLC7A5 378/4885CPB2 2555/4885CPB1 2381/4885
US-20240245796-A1 LINKERS, DRUG LINKERS AND CONJUGATES THEREOF AND METHODS OF USING THE SAME PAICS, DHFR, CD44 SLC7A5 378/4885CPB2 2555/4885CPB1 2381/4885
US-20220112234-A1 METHOD FOR PRODUCING PEPTIDE COMPOUND, PROTECTIVE GROUP-FORMING REAGENT, AND CONDENSED POLYCYCLIC COMPOUND C9, GRPR, VIP SLC7A5 2929/4885CPB2 803/4885CPB1 1295/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.