SCHEMBL7489509

SCHEMBL7489509

CCCCCCc1n[c]c2nc[nH]c2n1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 6/20 0.33
XDH P47989 2/20 0.33
KCNH2 Q12809 1/20 0.33
ADORA2B P29275 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
PAK1 Q13153 1/20 0.32
ADORA3 P0DMS8 1/20 0.31
ADORA2A P29274 1/20 0.31
ALDH1A1 P00352 1/20 0.31
PKM P14618 1/20 0.31
HPGD P15428 1/20 0.31
EPHX1 P07099 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7482351 0.98 GPR84 (0.34) GPR84XDHKCNH2ADORA2BCDK1
SCHEMBL7487571 0.94 HRH3 (0.34) XDHCDK1CCNB1HRH3ADORA3
SCHEMBL7496538 0.88 PDK2 (0.30)
SCHEMBL7493590 0.81
SCHEMBL7491723 0.78 CDK1 (0.39) XDHKCNH2ADORA2BCDK1CCNB1
SCHEMBL7490134 0.76 PAK1 (0.39) XDHCDK1CCNB1PAK1ADORA3
SCHEMBL8041008 0.71 HRH3 (0.36) XDHCDK1CCNB1HRH4HRH3
SCHEMBL7488939 0.71 ADORA3 (0.38) XDHCDK1CCNB1HRH3PAK1
SCHEMBL7542834 0.71 XDH (0.38) GPR84XDHKCNH2ALDH1A1PKM
SCHEMBL7488641 0.70 ADORA2A (0.34) GPR84XDHKCNH2ADORA2BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915093-B1 AMIDE DERIVATIVES OTSUKA PHARMA CO LTD (JP) 2002-11-27 EP disclosed
US-6166016-A Amide derivatives OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 2000-12-26 US disclosed
EP-0915093-A1 AMIDE DERIVATIVES OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1999-05-12 EP disclosed