SCHEMBL7490908

SCHEMBL7490908

O=CCc1cccc(Cc2c(F)cccc2F)c1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
DAO P14920 4/20 0.36
TDP1 Q9NUW8 2/20 0.34
AR P10275 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
PTPN1 P18031 1/20 0.33
LMNA P02545 1/20 0.33
TAAR1 Q96RJ0 2/20 0.32
ERN1 O75460 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12345478 0.79 MAOB (0.39) MEN1KMT2ALMNA
SCHEMBL1459660 0.78 ERN1 (0.40) KDM4EALDH1A1SMN1; SMN2DAOTDP1
SCHEMBL7083313 0.76 CALM1 (0.52) LMNA
SCHEMBL167999 0.74 TAAR1 (0.52) ALDH1A1SMN1; SMN2DAOTDP1LMNA
SCHEMBL13377016 0.71 DAO (0.50) KDM4EALDH1A1DAOMEN1KMT2A
SCHEMBL7497723 0.70 HRH3 (0.34) TAAR1
SCHEMBL26987979 0.70 MAOB (0.44) ALDH1A1LMNA
SCHEMBL7081270 0.70 IL4I1 (0.50) ALDH1A1SMN1; SMN2PTPN1LMNA
SCHEMBL7930766 0.70 MGLL (0.44) ALDH1A1SMN1; SMN2LMNATP53
SCHEMBL5500689 0.70 ALDH1A1 (0.44) ALDH1A1TDP1MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1196384-A4 1-(AROMATIC- OR HETEROAROMATIC-SUBSTITUTED)-3-(HETEROAROMATIC SUBSTITUTED)-1,3-PROPANEDIONES AND USES THEREOF MERCK & CO INC (US) 2002-10-23 EP disclosed
EP-1196384-A1 1-(AROMATIC- OR HETEROAROMATIC-SUBSTITUTED)-3-(HETEROAROMATIC SUBSTITUTED)-1,3-PROPANEDIONES AND USES THEREOF Merck & Co., Inc. (US) 2002-04-17 EP disclosed
WO-2001000578-A1 1-(AROMATIC- OR HETEROAROMATIC-SUBSTITUTED)-3-(HETEROAROMATIC SUBSTITUTED)-1,3-PROPANEDIONES AND USES THEREOF MERCK & CO., INC. (US) 2001-01-04 WO disclosed