SCHEMBL749653

SCHEMBL749653

CCCCOC(=O)NC(CCC(=O)OCc1ccccc1)C(=O)N(C)OC

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
MEN1 O00255 1/20 0.52
HPGD P15428 1/20 0.52
KMT2A Q03164 1/20 0.52
CCKBR P32239 2/20 0.51
CTSL P07711 2/20 0.48
CTSS P25774 2/20 0.48
SIRT2 Q8IXJ6 7/20 0.46
SIRT1 Q96EB6 7/20 0.46
SIRT3 Q9NTG7 3/20 0.46
CTSK P43235 3/20 0.45
BCHE P06276 1/20 0.44
ACHE P22303 1/20 0.44
CTSB P07858 1/20 0.44
CYP3A4 P08684 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18954330 0.86 ALDH1A1 (0.58) ALDH1A1MEN1HPGDKMT2ACCKBR
SCHEMBL16847591 0.86 CTSL (0.62) CTSLCTSSSIRT2SIRT1SIRT3
SCHEMBL18649575 0.85 CNR2 (0.48) ALDH1A1MEN1HPGDKMT2ACCKBR
SCHEMBL749652 0.85 SIRT2 (0.49) ALDH1A1MEN1HPGDKMT2ACTSL
SCHEMBL2300340 0.84 ALDH1A1 (0.56) ALDH1A1MEN1HPGDKMT2ACCKBR
SCHEMBL7293004 0.84 CTSK (0.51) ALDH1A1MEN1KMT2ACTSLCTSS
SCHEMBL13970298 0.84 CTSK (0.51) ALDH1A1MEN1KMT2ACTSLCTSS
SCHEMBL4961276 0.84 CTSK (0.57) ALDH1A1MEN1KMT2ACTSLCTSS
SCHEMBL13058656 0.84 CTSK (0.57) ALDH1A1MEN1KMT2ACTSLCTSS
SCHEMBL8219708 0.84 JAK3 (0.58) CCKBRCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430014-A1 ANTIVIRAL COMPOUNDS Gilead Sciences, Inc. (US) 2012-03-21 EP disclosed
WO-2010132601-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2010-11-18 WO disclosed