SCHEMBL7500754

SCHEMBL7500754

CCCC(c1ccccc1)N1CCC(Nc2ccccc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 7/20 0.51
OPRD1 P41143 7/20 0.51
OPRK1 P41145 7/20 0.51
OPRL1 P41146 7/20 0.51
CARM1 Q86X55 1/20 0.48
PRMT6 Q96LA8 1/20 0.48
KDM4E B2RXH2 1/20 0.40
DPP4 P27487 1/20 0.40
SLC6A4 P31645 1/20 0.40
ALDH1A1 P00352 1/20 0.39
CCR6 P51684 1/20 0.39
MC4R P32245 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9523741 0.78 OPRM1 (0.55) OPRM1OPRD1OPRK1OPRL1CARM1
SCHEMBL28738958 0.78 CYP2D6 (0.59) OPRM1OPRD1OPRK1OPRL1CARM1
SCHEMBL10598753 0.77 OPRM1 (0.63) OPRM1OPRD1OPRK1OPRL1SLC6A4
SCHEMBL20205982 0.77 CARM1 (0.52) CARM1PRMT6KDM4EALDH1A1CCR6
SCHEMBL7405479 0.76 OPRK1 (0.52) OPRM1OPRD1OPRK1OPRL1SLC6A4
SCHEMBL11447302 0.76 ALDH1A1 (0.61) CARM1PRMT6ALDH1A1CCR6
SCHEMBL10601133 0.76 CYP1A2 (0.62) OPRM1OPRD1OPRK1OPRL1SLC6A4
SCHEMBL113896 0.76 CYP1A2 (0.62) OPRM1OPRD1OPRK1OPRL1SLC6A4
SCHEMBL25103860 0.74 CARM1 (0.47) CARM1PRMT6KDM4EALDH1A1CCR6
SCHEMBL12513620 0.74 MC4R (0.65) OPRM1OPRD1OPRK1OPRL1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1265870-A1 NEW CCR5 MODULATORS: BENZIMIDAZOLES OR BENZOTRIAZOLES AstraZeneca AB (SE) 2002-12-18 EP disclosed
WO-2001066525-A1 NEW CCR5 MODULATORS: BENZIMIDAZOLES OR BENZOTRIAZOLES ASTRAZENECA AB (SE) 2001-09-13 WO disclosed