SCHEMBL7510667

SCHEMBL7510667

O[C@@H]([C@H](O)[C@@H](COCc1ccccc1F)OCc1cccs1)[C@@H](COCc1ccccc1F)OCc1ccc(F)cc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.39
HPGD P15428 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TSHR P16473 1/20 0.36
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
EGFR P00533 1/20 0.34
TOP2A P11388 1/20 0.34
TOP2B Q02880 1/20 0.34
POLB P06746 2/20 0.34
SLC1A3 P43003 1/20 0.34
SLC1A2 P43004 1/20 0.34
SLC1A1 P43005 1/20 0.34
HSP90AA1 P07900 1/20 0.34
MAPK1 P28482 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.32
SLC6A3 Q01959 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7511715 0.89 NPSR1 (0.41) NPSR1HPGDTSHRALDH1A1GAA
SCHEMBL7989987 0.89 NPSR1 (0.46) NPSR1HPGDSMN1; SMN2TSHRALDH1A1
SCHEMBL7987648 0.89 HSP90AA1 (0.39) SMN1; SMN2ALDH1A1GAAHSP90AA1KDM4E
SCHEMBL7987303 0.86 HSP90AA1 (0.43) SMN1; SMN2ALDH1A1GAAHSP90AA1KDM4E
SCHEMBL7447822 0.85 HSP90AA1 (0.44) GAAHSP90AA1MAPK1KDM4E
SCHEMBL7450924 0.85 NPSR1 (0.39) NPSR1HPGDTSHRALDH1A1GAA
SCHEMBL7989824 0.81 ALDH1A1 (0.39) NPSR1ALDH1A1GAAKDM4EMAPT
SCHEMBL7989289 0.81 CA1 (0.42) TSHRALDH1A1GAAHSP90AA1MAPK1
SCHEMBL7989311 0.80 CA1 (0.44) TSHRALDH1A1GAASLC1A1HSP90AA1
SCHEMBL7517976 0.80 ALDH1A1 (0.45) HPGDSMN1; SMN2TSHRALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1175385-A1 D-MANNITOL DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS Pharmacor Inc. (CA) 2002-01-30 EP disclosed
US-6313177-B1 AS ANTIVIRAL AGENTS PHARMACOR INC. (CA) 2001-11-06 US disclosed
WO-2000066524-A1 D-MANNITOL DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS PHARMACOR INC. (CA) 2000-11-09 WO disclosed