SCHEMBL7511039

SCHEMBL7511039

Cc1cccc(-c2c(-c3ccc(S(C)(=O)=O)cc3)nc(C(F)(F)F)n2COCC[Si](C)(C)C)c1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.48
PTGS1 P23219 4/20 0.48
DGAT1 O75907 2/20 0.39
SDHB P21912 1/20 0.39
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7136177 0.86 PTGS2 (0.44) PTGS2PTGS1DGAT1
SCHEMBL7087803 0.77 PTGS2 (0.45) PTGS2PTGS1
SCHEMBL8802398 0.69 ALOX5AP (0.38) PTGS2PTGS1DGAT1
SCHEMBL16069684 0.68 PTGS2 (0.36) PTGS2PTGS1NR1H2NR1H3
SCHEMBL2148593 0.68 CYP1A2 (0.43)
SCHEMBL2315531 0.67 DGAT1 (0.35) DGAT1NR1H2NR1H3
SCHEMBL7087564 0.66 MAPK14 (0.58) PTGS2PTGS1SDHB
SCHEMBL19952994 0.66 PTGS2 (0.58) PTGS2PTGS1SDHB
SCHEMBL2148279 0.66 PIN1 (0.41)
SCHEMBL14701092 0.66 PDE4D (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0772601-B1 4,5-SUBSTITUTED IMIDAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2002-09-18 EP disclosed
US-6426360-B1 ANTIARTHRITIC AGENTS G D SEARLE & CO. 2002-07-30 US disclosed
WO-1996003387-A1 4,5-SUBSTITUTED IMIDAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-02-08 WO disclosed