SCHEMBL7512573

SCHEMBL7512573

CCCCC1(CCCC)C(=O)Sc2cc(OCC(=O)O)c(OC)cc2N(c2ccccc2)C1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 2/20 0.44
ALDH1A1 P00352 5/20 0.42
NPSR1 Q6W5P4 2/20 0.42
GPR55 Q9Y2T6 2/20 0.42
SLC10A2 Q12908 1/20 0.40
CYP2C19 P33261 1/20 0.39
KDM4E B2RXH2 3/20 0.39
HPGD P15428 2/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
PKM P14618 1/20 0.38
SMN1; SMN2 Q16637 6/20 0.38
POLB P06746 3/20 0.38
LMNA P02545 4/20 0.38
HTT P42858 2/20 0.38
CNR1 P21554 1/20 0.38
MEN1 O00255 6/20 0.37
KMT2A Q03164 6/20 0.37
MAPT P10636 2/20 0.37
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6993131 0.91 ELANE (0.41) ELANEALDH1A1NPSR1GPR55CYP2C19
Ethyl Bromo Acetate SCHEMBL7509727 0.88 ALDH1A1 (0.39) ELANEALDH1A1NPSR1GPR55CYP2C19
SCHEMBL6993818 0.88 ELANE (0.43) ELANEALDH1A1NPSR1GPR55CYP2C19
SCHEMBL6987940 0.86 ELANE (0.48) ELANEALDH1A1NPSR1GPR55SLC10A2
SCHEMBL6993226 0.80 ELANE (0.41) ELANEALDH1A1CYP2C19KDM4EHPGD
SCHEMBL6992850 0.79 ELANE (0.40) ELANEALDH1A1NPSR1GPR55PKM
SCHEMBL7507444 0.78 ELANE (0.45) ELANEALDH1A1NPSR1GPR55CYP2C19
SCHEMBL6987548 0.78 ELANE (0.47) ELANEALDH1A1NPSR1GPR55CYP2C19
Water SCHEMBL7515031 0.77 ELANE (0.45) ELANEALDH1A1NPSR1GPR55CYP2C19
SCHEMBL6992847 0.76 ELANE (0.43) ELANEALDH1A1NPSR1GPR55CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244621-A1 NITRILE DERIVATIVES AS CATHEPSIN K INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2002-10-02 EP disclosed
WO-2001047886-A1 NITRILE DERIVATIVES AS CATHEPSIN K INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2001-07-05 WO disclosed