SCHEMBL7513532

SCHEMBL7513532

CC(=O)O[C@@H]1OCC[C@@H]1NC(=O)[C@H](CC(C)C)NC(=O)c1cnc2ccccc2c1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 6/20 0.61
CAPNS1 P04632 2/20 0.60
CASP1 P29466 1/20 0.49
CASP3 P42574 1/20 0.49
CTSK P43235 6/20 0.48
CCR1 P32246 6/20 0.48
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7510995 0.89 CAPN1 (0.49) CAPN1CAPNS1CCR1
SCHEMBL7515201 0.87 CAPN1 (0.59) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL7515061 0.85 CTSK (0.59) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL8810074 0.81 CAPN1 (0.66) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL8810052 0.81 CAPN1 (0.66) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL8404224 0.80 CAPN1 (0.65) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL8404221 0.80 CAPN1 (0.65) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL7517376 0.80 CAPN1 (0.65) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL8808955 0.79 CAPN1 (0.62) CAPN1CAPNS1CASP1CCR1
SCHEMBL8808938 0.79 CAPN1 (0.62) CAPN1CAPNS1CASP1CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP claimed
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP disclosed