SCHEMBL7515201

SCHEMBL7515201

CC(C)C[C@H](NC(=O)c1cnc2ccccc2c1)C(=O)N[C@H]1CCOC1O

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 14/20 0.59
CAPNS1 P04632 3/20 0.57
CASP1 P29466 1/20 0.54
CASP3 P42574 1/20 0.54
CCR1 P32246 4/20 0.49
CTSK P43235 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7514760 0.88 CAPN1 (0.49) CAPN1CAPNS1CCR1
SCHEMBL7513532 0.87 CAPN1 (0.61) CAPN1CAPNS1CASP1CASP3CCR1
SCHEMBL8812460 0.86 CASP1 (0.72) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL8812453 0.86 CASP1 (0.72) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL8809577 0.84 CAPN1 (0.71) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL8809563 0.84 CAPN1 (0.71) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL7517851 0.83 CTSK (0.63) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL8810040 0.79 CAPN1 (0.70) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL8810031 0.79 CAPN1 (0.70) CAPN1CAPNS1CASP1CASP3CTSK
SCHEMBL8408034 0.79 CAPN1 (0.71) CAPN1CAPNS1CASP1CASP3CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP claimed
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP disclosed