SCHEMBL7514760

SCHEMBL7514760

O=C(N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCOC1O)c1cnc2ccccc2c1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 6/20 0.49
CCR1 P32246 1/20 0.46
CAPNS1 P04632 1/20 0.44
CCKBR P32239 1/20 0.43
MC4R P32245 2/20 0.43
CXCR4 P61073 1/20 0.43
HPGDS O60760 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7515201 0.88 CAPN1 (0.59) CAPN1CCR1CAPNS1
SCHEMBL7510995 0.87 CAPN1 (0.49) CAPN1CCR1CAPNS1CCKBRMC4R
SCHEMBL7514607 0.83 CAPN1 (0.49) CAPN1CCR1
SCHEMBL7513532 0.75 CAPN1 (0.61) CAPN1CCR1CAPNS1
SCHEMBL7514977 0.75 CAPN1 (0.59) CAPN1CAPNS1
SCHEMBL7514986 0.74 CAPN1 (0.52) CAPN1CAPNS1
SCHEMBL8812581 0.74 CTSK (0.60) CAPN1
SCHEMBL8812573 0.74 CTSK (0.60) CAPN1
SCHEMBL8812460 0.73 CASP1 (0.72) CAPN1CAPNS1
SCHEMBL8812453 0.73 CASP1 (0.72) CAPN1CAPNS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP claimed
EP-0641800-B1 Lactol derivatives as inhibitors of cathepsin L TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-01-16 EP disclosed