SCHEMBL7516105

SCHEMBL7516105

Cc1cc2c(O)cccc2nc1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
HPGD P15428 3/20 0.48
GAA P10253 3/20 0.48
KDM4E B2RXH2 1/20 0.48
STAT3 P40763 1/20 0.48
GPR3 P46089 1/20 0.44
HSD17B1 P14061 1/20 0.42
HSD17B2 P37059 1/20 0.42
ACHE P22303 1/20 0.42
CYP1A2 P05177 4/20 0.41
ERN1 O75460 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
UHRF1 Q96T88 1/20 0.41
HTT P42858 2/20 0.40
NUDT1 P36639 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PDE10A Q9Y233 1/20 0.40
BACE1 P56817 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL862361 0.82 PDE3B (0.49) ALDH1A1HPGDGPR3CYP1A2OPRM1
SCHEMBL27600483 0.81 ALDH1A1 (0.46) ALDH1A1HPGDGAAKDM4ESTAT3
SCHEMBL19700637 0.77 GPR3 (0.44) ALDH1A1HPGDGAAKDM4ESTAT3
SCHEMBL28042222 0.77 ALDH1A1 (0.56) ALDH1A1HPGDGAAKDM4EGPR3
SCHEMBL29923623 0.77 BACE1 (0.47) ALDH1A1HPGDGAAKDM4ESTAT3
SCHEMBL24916325 0.77 BACE1 (0.47) ALDH1A1HPGDGAAKDM4ESTAT3
SCHEMBL15119531 0.77 ALDH1A1 (0.58) ALDH1A1HPGDGAAKDM4ESTAT3
SCHEMBL28073764 0.77 PDE10A (0.47) ALDH1A1HPGDKDM4EHSD17B10PDE10A
SCHEMBL24915591 0.74 DHFR (0.48) ALDH1A1HPGDGPR3CYP1A2OPRM1
SCHEMBL28492152 0.74 KDM4E (0.47) ALDH1A1HPGDGAAKDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101747336-B Novel method for synthesizing Repirinast JIANGSU JUMPCAN MEDICINES CO LTD 2012-07-18 CN claimed
CN-101747336-A Novel method for synthesizing Repirinast JIANGSU JUMPCAN MEDICINES CO L 2010-06-23 CN claimed
CN-101747336-B Novel method for synthesizing Repirinast JIANGSU JUMPCAN MEDICINES CO LTD 2012-07-18 CN disclosed
CN-101316591-B Quinoline compound and pharmaceutical application thereof ARGENTA ORAL THERAPEUTICS LTD. (GB) 2012-02-01 CN disclosed
CN-101747336-A Novel method for synthesizing Repirinast JIANGSU JUMPCAN MEDICINES CO L 2010-06-23 CN disclosed
CN-101316591-A Quinolines and their therapeutic use ARGENTA DISCOVERY LTD (GB) 2008-12-03 CN disclosed
WO-1995021825-A1 6-ARYL-(METHYL- OR METHYLIDONE)-QUINOLINE DERIVATIVES AS VOLTAGE-GATED POTASSIUM CHANNEL BLOCKERS JOHN WYETH & BROTHER LTD. (GB) 1995-08-17 WO disclosed
EP-0363212-A2 Novel heterocyclic compounds and anticancer-drug reinforcing agents containing them as effective components MITSUI TOATSU CHEMICALS, Inc. (JP) 1990-04-11 EP disclosed