SCHEMBL7516495

SCHEMBL7516495

N=C(Nc1ccc2c(c1)CN(CCO)CCC2)C1=CC=CCC1=S

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
KDM4E B2RXH2 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
ADRA2A P08913 2/20 0.34
ALOX15 P16050 2/20 0.34
TP53 P04637 1/20 0.34
BTK Q06187 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
POLB P06746 1/20 0.34
USP2 O75604 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
GAA P10253 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPK1 P28482 1/20 0.33
ACVR1 Q04771 1/20 0.33
LMNA P02545 2/20 0.32
HSD17B10 Q99714 1/20 0.32
CREBBP Q92793 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7512685 0.94 BTK (0.38) ALDH1A1KDM4EBTKHTTUSP2
SCHEMBL7824786 0.86 DRD2 (0.37) ALDH1A1KDM4EALOX15TP53HTT
SCHEMBL7827942 0.84 DRD2 (0.45) ALDH1A1KDM4ESMN1; SMN2ALOX15TP53
SCHEMBL7818532 0.84 L3MBTL3 (0.38) KDM4ESMN1; SMN2BTKHTTPOLB
SCHEMBL7827664 0.83 ROCK2 (0.38) KDM4E
SCHEMBL7829164 0.78 HRH3 (0.35) ALDH1A1KDM4EBTKUSP2RXFP1
SCHEMBL7512428 0.76 L3MBTL3 (0.31)
SCHEMBL7510864 0.75
SCHEMBL7480136 0.75 MAPT (0.33) ALDH1A1KDM4ESMN1; SMN2TP53HPGD
SCHEMBL7515406 0.75 LMNA (0.48) ALDH1A1KDM4ESMN1; SMN2TP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861250-B1 AMIDINE AND ISOTHIOUREA DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2002-02-13 EP claimed