SCHEMBL7512685

SCHEMBL7512685

N=C(Nc1ccc2c(c1)CN(CCO)CC2)C1=CC=CCC1=S

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.38
ACVR1 Q04771 1/20 0.36
GAA P10253 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PRMT5 O14744 4/20 0.35
WDR77 Q9BQA1 4/20 0.35
JAK2 O60674 2/20 0.35
FLT3 P36888 2/20 0.35
USP2 O75604 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
WEE1 P30291 1/20 0.34
DRD2 P14416 2/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
ABCB1 P08183 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7516495 0.94 ALDH1A1 (0.36) BTKACVR1GAAMEN1KMT2A
SCHEMBL7824786 0.92 DRD2 (0.37) GAAITGB3ITGA2BMEN1KMT2A
SCHEMBL7827942 0.90 DRD2 (0.45) GAAITGB3ITGA2BMEN1KMT2A
SCHEMBL7818532 0.90 L3MBTL3 (0.38) BTKGAAITGB3ITGA2BMEN1
SCHEMBL7827664 0.87 ROCK2 (0.38) DRD2KDM4E
SCHEMBL7829164 0.81 HRH3 (0.35) BTKUSP2ALDH1A1KDM4E
SCHEMBL7512428 0.77 L3MBTL3 (0.31)
SCHEMBL7510864 0.77
SCHEMBL7480136 0.77 MAPT (0.33) GAAMEN1KMT2AALDH1A1KDM4E
SCHEMBL7517482 0.76 MAOA (0.40) KMT2AMAPTHTTPLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861250-B1 AMIDINE AND ISOTHIOUREA DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2002-02-13 EP claimed