SCHEMBL7517537

SCHEMBL7517537

CCCC1c2cc(NC(=N)C3=CC=CCC3=S)ccc2CCN1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN2 Q9H2S1 4/20 0.33
KCNN3 Q9UGI6 4/20 0.33
KCNN1 Q92952 2/20 0.33
HTR1A P08908 2/20 0.33
OPRK1 P41145 2/20 0.33
NR1I2 O75469 1/20 0.33
MAOA P21397 1/20 0.33
PTGS2 P35354 1/20 0.33
SLC6A3 Q01959 1/20 0.33
TP53 P04637 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
DRD2 P14416 2/20 0.32
DRD4 P21917 1/20 0.32
CTSS P25774 1/20 0.31
OPRM1 P35372 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7517482 0.85 MAOA (0.40) HTR1AMAOACTSSHTR2AHTR7
SCHEMBL7512989 0.79 F2 (0.41) KDM4EALDH1A1DRD2DRD4OPRM1
SCHEMBL7824786 0.78 DRD2 (0.37) HTR1ATP53KDM4EALDH1A1ALOX15
SCHEMBL7827664 0.77 ROCK2 (0.38) MAOAKDM4EDRD2
SCHEMBL7827942 0.77 DRD2 (0.45) TP53MAPK1KDM4EALDH1A1ALOX15
SCHEMBL7510363 0.76 CNR1 (0.41) CTSS
SCHEMBL7516949 0.76 NPC1 (0.41) HTR1AMAPK1KDM4EALDH1A1HSD17B10
SCHEMBL7818532 0.76 L3MBTL3 (0.38) KDM4EDRD2DRD1POLB
SCHEMBL7521473 0.75 CNR1 (0.41)
SCHEMBL7506683 0.75 F2 (0.42) KDM4EALDH1A1DRD2DRD4OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861250-B1 AMIDINE AND ISOTHIOUREA DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2002-02-13 EP claimed