SCHEMBL7517609

SCHEMBL7517609

CN(C)c1ccc([Si](C)(C)CCc2cc(C(C)(C)C)c(OC(=O)CCC(=O)O)c(C(C)(C)C)c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 10/20 0.45
GAA P10253 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
ALOX15 P16050 1/20 0.31
NFKB1 P19838 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
MCL1 Q07820 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CALM1 P0DP23 1/20 0.31
LTB4R Q15722 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7521009 0.91 VCAM1 (0.37) VCAM1GAAALOX15CALM1
SCHEMBL7522609 0.86 CALM1 (0.33) VCAM1GAAALDH1A1MAPTCALM1
SCHEMBL7518758 0.84 VCAM1 (0.47) VCAM1LTB4R
SCHEMBL7527917 0.80 VCAM1 (0.40) VCAM1GAAALOX15
SCHEMBL7522270 0.77 GAA (0.37) VCAM1GAA
SCHEMBL7525872 0.76 VCAM1 (0.36) VCAM1GAAALDH1A1MAPK1LTB4R
SCHEMBL7524217 0.74 VCAM1 (0.37) VCAM1GAAALDH1A1MAPTRAB9A
SCHEMBL7523700 0.73 NR1H4 (0.35) VCAM1GAA
SCHEMBL7523688 0.72 VCAM1 (0.35) VCAM1GAAALDH1A1MAPT
SCHEMBL7523462 0.71 VCAM1 (0.52) VCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900225-B1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS AVENTIS PHARMA INC (US) 2002-01-30 EP disclosed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US disclosed