SCHEMBL7523700

SCHEMBL7523700

CC(=O)Oc1c(C(C)(C)C)cc(CC[Si](C)(C)c2ccc(N)cc2)cc1C(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.35
CYP19A1 P11511 1/20 0.33
ESRRG P62508 1/20 0.33
GAA P10253 3/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
EPHX2 P34913 1/20 0.32
VCAM1 P19320 4/20 0.32
KMT2A Q03164 2/20 0.31
PPIB P23284 1/20 0.31
PPIA P62937 1/20 0.31
PPID Q08752 1/20 0.31
PPIG Q13427 1/20 0.31
MEN1 O00255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7516554 0.86 GAA (0.34) NR1H4GAAVCAM1KMT2AMEN1
SCHEMBL7522609 0.86 CALM1 (0.33) NR1H4GAAVCAM1KMT2AMEN1
SCHEMBL7518915 0.81 GAA (0.43) GAAKMT2AMEN1
SCHEMBL7520189 0.80 VCAM1 (0.37) NR1H4CYP19A1CTSLCTSBVCAM1
SCHEMBL7522270 0.76 GAA (0.37) GAAVCAM1KMT2AMEN1
SCHEMBL7527917 0.74 VCAM1 (0.40) GAAVCAM1KMT2APPIDMEN1
SCHEMBL9354087 0.74 VCAM1 (0.45) GAAVCAM1KMT2A
SCHEMBL7521009 0.73 VCAM1 (0.37) GAAVCAM1KMT2A
SCHEMBL7517609 0.73 VCAM1 (0.45) GAAVCAM1
SCHEMBL4324980 0.73 NR1H4 (0.39) NR1H4CYP19A1VCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900225-B1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS AVENTIS PHARMA INC (US) 2002-01-30 EP disclosed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US disclosed