Metitepine

Metitepine

SCHEMBL7517783

CSc1ccc2c(c1)[C@H](N1CCN(C)CC1)Cc1ccccc1S2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 4/20 1.00
MAPT P10636 4/20 1.00
TP53 P04637 4/20 1.00
CYP3A4 P08684 4/20 1.00
SMN1; SMN2 Q16637 3/20 1.00
CYP1A2 P05177 3/20 1.00
CYP2D6 P10635 3/20 1.00
HTR2C P28335 3/20 1.00
HTR1A P08908 2/20 1.00
HTR2A P28223 2/20 1.00
TDP1 Q9NUW8 2/20 1.00
NPC1 O15118 2/20 1.00
MTOR P42345 2/20 1.00
RAB9A P51151 2/20 1.00
CYP2C19 P33261 2/20 1.00
ALDH1A1 P00352 1/20 1.00
HTT P42858 1/20 1.00
HTR5A P47898 1/20 1.00
HTR6 P50406 1/20 1.00
CYP2C9 P11712 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Metitepine SCHEMBL113526 1.00 HTR7 (1.00) HTR7MAPTTP53CYP3A4SMN1; SMN2
Metitepine SCHEMBL14359602 1.00 HTR7 (1.00) HTR7MAPTTP53CYP3A4SMN1; SMN2
Metitepine SCHEMBL29496251 1.00 HTR7 (1.00) HTR7MAPTTP53CYP3A4SMN1; SMN2
Metitepine SCHEMBL8169076 0.94 HTR7 (0.89) HTR7MAPTTP53CYP3A4SMN1; SMN2
Metitepine SCHEMBL466985 0.92 MAPT (1.00) HTR7MAPTTP53CYP3A4SMN1; SMN2
Metitepine SCHEMBL31360614 0.92 MAPT (1.00) HTR7MAPTTP53CYP3A4SMN1; SMN2
Metitepine SCHEMBL15475310 0.91 MAPT (1.00) HTR7MAPTTP53CYP3A4SMN1; SMN2
Metitepine SCHEMBL2048660 0.91 MAPT (1.00) HTR7MAPTTP53CYP3A4SMN1; SMN2
SCHEMBL8877190 0.88 MAPT (0.79) HTR7MAPTTP53CYP3A4SMN1; SMN2
SCHEMBL11876604 0.87 HTR7 (0.77) HTR7MAPTTP53CYP3A4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240165079-A1 COMBINATION PRODUCT FOR THE TREATMENT OF NEUROLOGICAL AND/OR PSYCHIATRIC DISORDERS CONSEJO SUPERIOR INVESTIGACION (ES) 2024-05-23 US disclosed
US-20240115564-A1 HTR1F ANTAGONISTS FOR IMPROVEMENT OF BETA CELL SURVIVAL AND FUNCTION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-04-11 US disclosed
US-20230330063-A1 COMBINATION PRODUCT FOR THE TREATMENT OF NEUROLOGICAL AND/OR PSYCHIATRIC DISORDERS CONSEJO SUPERIOR INVESTIGACION (ES) 2023-10-19 US disclosed
US-11723894-B2 Combination product for the treatment of neurological and/or psychiatric disorders TERRAN BIOSCIENCES, INC. (US) 2023-08-15 US disclosed
WO-2022155152-A1 HTR1F ANTAGONISTS FOR IMPROVEMENT OF BETA CELL SURVIVAL AND FUNCTION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-07-21 WO disclosed
US-20200397752-A1 COMBINATION PRODUCT FOR THE TREATMENT OF NEUROLOGICAL AND/OR PSYCHIATRIC DISORDERS Consejo Superior de Investigacions Cientificas (CSIS) (ES) 2020-12-24 US disclosed
EP-3713568-A1 COMBINATION PRODUCT FOR THE TREATMENT OF NEUROLOGICAL AND/OR PSYCHIATRIC DISORDERS Consejo Superior de Investigaciones Cientificas (CSIC) (ES) 2020-09-30 EP disclosed
US-20020182594-A1 Chemomagnetic retrieval of CMV and CMV infected cells CHEMOCENTRYX (US) 2002-12-05 US disclosed
US-20020127544-A1 Modulators of US 28 CHEMOCENTRYX 2002-09-12 US disclosed
WO-2002062956-A2 CHEMOMAGNETIC RETRIEVAL OF CMV AND CMV INFECTED CELLS CHEMOCENTRYX, INC. (US) 2002-08-15 WO disclosed
WO-2002017900-A2 MODULATORS OF US28 (CHEMOKINES) FOR TREATING CYTOMEGALOVIRUS INFECTIONS CHEMOCENTRYX, INC. (US) 2002-03-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200397752-A1 COMBINATION PRODUCT FOR THE TREATMENT OF NEUROLOGICAL AND/OR PSYCHIATRIC DISORDERS HTR2A, HTR2C, HTR1A HTR7 11/4885MAPT 322/4885TP53 4651/4885
US-20230330063-A1 COMBINATION PRODUCT FOR THE TREATMENT OF NEUROLOGICAL AND/OR PSYCHIATRIC DISORDERS HTR2A, HTR2C, HTR1A HTR7 12/4885MAPT 300/4885TP53 4645/4885
US-20240115564-A1 HTR1F ANTAGONISTS FOR IMPROVEMENT OF BETA CELL SURVIVAL AND FUNCTION HTR1F, HTR1D, HTR1E HTR7 16/4885MAPT 4647/4885TP53 3093/4885
US-20020127544-A1 Modulators of US 28 CCR8, CCL5, CXCL10 HTR7 2029/4885MAPT 4038/4885TP53 590/4885
US-20240165079-A1 COMBINATION PRODUCT FOR THE TREATMENT OF NEUROLOGICAL AND/OR PSYCHIATRIC DISORDERS HTR2A, HTR2C, HTR1A HTR7 11/4885MAPT 322/4885TP53 4651/4885
US-11723894-B2 Combination product for the treatment of neurological and/or psychiatric disorders HTR2A, HTR2C, HTR1A HTR7 11/4885MAPT 322/4885TP53 4651/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.