SCHEMBL7523485

SCHEMBL7523485

CC(=O)Oc1cc(C)c(SC[Si](C)(C)c2ccc(N)cc2)c(C)c1C

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.40
HTT P42858 1/20 0.36
PTPN1 P18031 2/20 0.34
CYP19A1 P11511 1/20 0.33
ACHE P22303 1/20 0.32
PTGS2 P35354 2/20 0.31
CTSL P07711 1/20 0.30
CTSB P07858 1/20 0.30
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7525047 0.79 TSHR (0.34) HTT
SCHEMBL7520189 0.72 VCAM1 (0.37) CYP19A1CTSLCTSB
SCHEMBL7521661 0.66 KDM4E (0.31) ALDH1A1
SCHEMBL1469593 0.63 ACHE (0.59) POLBHTTCYP19A1ACHEALDH1A1
SCHEMBL4520980 0.63 ACHE (0.46) POLBHTTCYP19A1ACHEALDH1A1
SCHEMBL2910532 0.62 POLB (0.62) POLBHTTPTPN1ACHEALDH1A1
SCHEMBL7519795 0.62 HTT (0.49) POLBHTTPTPN1PTGS2ALDH1A1
SCHEMBL7523700 0.61 NR1H4 (0.35) CYP19A1CTSLCTSB
SCHEMBL7520501 0.61 HTT (0.48) POLBHTTPTPN1ACHEPTGS2
SCHEMBL15642113 0.61 POLB (0.65) POLBHTTPTPN1ACHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900225-B1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS AVENTIS PHARMA INC (US) 2002-01-30 EP disclosed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US disclosed