SCHEMBL7524936

SCHEMBL7524936

CC(C)(C)c1cc(OC[Si](C)(C)c2ccccc2)ccc1OC(=O)CCC(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 4/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
RBP4 P02753 3/20 0.34
SQLE Q14534 1/20 0.34
PPARG P37231 1/20 0.33
PPARD Q03181 1/20 0.33
PPARA Q07869 1/20 0.33
ATM Q13315 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
ELANE P08246 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
FFAR1 O14842 2/20 0.32
FFAR4 Q5NUL3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7523462 0.87 VCAM1 (0.52) VCAM1NPSR1RBP4SQLE
SCHEMBL7525820 0.86 MAPT (0.38) PTGDR2MEN1KMT2ASQLEATM
SCHEMBL8517276 0.82 ADORA3 (0.35) PTGDR2MEN1KMT2ASQLEATM
SCHEMBL6054926 0.81 VCAM1 (0.51) VCAM1NPSR1KMT2AATMMAPT
Butyric Acid SCHEMBL27516493 0.79 ATM (0.42) NPSR1SQLEATMPOLBMAPT
SCHEMBL7526551 0.78 VCAM1 (0.41) VCAM1SQLE
Propionic Acid SCHEMBL27515791 0.77 POLB (0.44) NPSR1SQLEATMPOLBMAPT
SCHEMBL7525872 0.77 VCAM1 (0.36) VCAM1PTGDR2NPSR1RBP4
SCHEMBL7515882 0.76 ESRRA (0.45) NPSR1SQLEATMTDP1CYP2C9
SCHEMBL7518758 0.76 VCAM1 (0.47) VCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900225-A1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1999-03-10 EP claimed
WO-1997041129-A1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1997-11-06 WO claimed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US claimed
EP-0900225-B1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS AVENTIS PHARMA INC (US) 2002-01-30 EP disclosed
EP-0900225-A1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1999-03-10 EP disclosed
WO-1997041129-A1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1997-11-06 WO disclosed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US disclosed