SCHEMBL7525820

SCHEMBL7525820

CC(=O)Oc1ccc(OC[Si](C)(C)c2ccccc2)cc1C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.38
MAPK1 P28482 1/20 0.38
NR1H4 Q96RI1 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SQLE Q14534 1/20 0.36
KDM4E B2RXH2 3/20 0.35
TDP1 Q9NUW8 2/20 0.35
ATM Q13315 1/20 0.35
PTPN1 P18031 2/20 0.35
ALDH1A1 P00352 2/20 0.35
TSHR P16473 2/20 0.35
ELANE P08246 1/20 0.35
ESR1 P03372 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
HMGB1 P09429 1/20 0.35
HPGD P15428 1/20 0.35
GGT1 P19440 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517276 0.94 ADORA3 (0.35) MAPTMAPK1NR1H4PTGDR2MEN1
SCHEMBL7516405 0.86 KDM4E (0.40) MAPTMAPK1NR1H4PTGDR2KDM4E
SCHEMBL7524936 0.86 VCAM1 (0.40) MAPTPTGDR2MEN1KMT2ASQLE
SCHEMBL7523672 0.85 BACE1 (0.39) MAPTSQLEELANECYP3A4
SCHEMBL7515882 0.80 ESRRA (0.45) MAPTNR1H4SQLETDP1ATM
Propionic Acid SCHEMBL27515791 0.79 POLB (0.44) MAPTNR1H4SQLEATMALDH1A1
SCHEMBL5692389 0.77 CA2 (0.45) MAPTMAPK1MEN1KMT2ASQLE
Dimethylamine SCHEMBL7525639 0.77 ESRRA (0.43) MAPTNR1H4SQLETDP1ATM
SCHEMBL7524096 0.76 VCAM1 (0.38) MAPTKMT2ASQLEELANERAB9A
Butyric Acid SCHEMBL27516493 0.76 ATM (0.42) MAPTNR1H4SQLEATMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900225-A1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1999-03-10 EP claimed
WO-1997041129-A1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS HOECHST MARION ROUSSEL, INC. (US) 1997-11-06 WO claimed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US claimed
EP-0900225-B1 ALKYL-4-SILYL-PHENOLS AND ESTERS THEREOF AS ANTIATHEROSCLEROTIC AGENTS AVENTIS PHARMA INC (US) 2002-01-30 EP disclosed
US-5608095-A Alkyl-4-silyl-phenols and esters thereof as antiatherosclerotic agents HOECHST MARION ROUSSEL, INC. (US) 1997-03-04 US disclosed