SCHEMBL7525447

SCHEMBL7525447

CC(=O)NCC(=O)Cc1ccccc1-c1ccccn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.40
ALDH1A1 P00352 4/20 0.39
BRD4 O60885 1/20 0.39
BRD2 P25440 1/20 0.39
BRD3 Q15059 1/20 0.39
BAZ2B Q9UIF8 1/20 0.39
BAZ2A Q9UIF9 1/20 0.39
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
MTNR1A P48039 3/20 0.37
MTNR1B P49286 2/20 0.37
HPGDS O60760 2/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
P2RX7 Q99572 1/20 0.36
JAK1 P23458 1/20 0.35
TYK2 P29597 1/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28139433 0.79 BRD4 (0.39) ADORA2AALDH1A1BRD4BRD2BRD3
SCHEMBL7976970 0.77 ALDH1A1 (0.50) ADORA2AALDH1A1BRD4BRD2BRD3
SCHEMBL1177969 0.76 KDM4E (0.53) BRD4BRD2BRD3BAZ2BBAZ2A
SCHEMBL4777973 0.72 KDM4E (0.50) ADORA2AALDH1A1BRD4KDM4EPKM
SCHEMBL28958350 0.70 TGFBR1 (0.43) ADORA2AALDH1A1BRD4BRD2BRD3
SCHEMBL22230614 0.70 CHRNB2 (0.49) ALDH1A1BRD4BRD2BRD3BAZ2B
SCHEMBL477370 0.69 KDM4E (0.50) ALDH1A1BRD4KDM4EPKMHPGD
SCHEMBL24889874 0.69 KDM4E (0.38) ADORA2AALDH1A1BRD4BRD2BRD3
SCHEMBL21666537 0.69 KDM4E (0.54) ALDH1A1KDM4EPKMHPGDLMNA
SCHEMBL24888335 0.69 KDM4E (0.54) ALDH1A1KDM4EPKMHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0983228-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-08-07 EP disclosed
EP-0983228-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-03-08 EP disclosed
WO-1998050342-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1998-11-12 WO disclosed