SCHEMBL7528375

SCHEMBL7528375

C1=CN(c2cccnc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
CHRNB2 P17787 9/20 0.45
CHRNA4 P43681 9/20 0.45
CHRNB4 P30926 5/20 0.44
CHRNA3 P32297 5/20 0.44
CHRNA7 P36544 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2A6 P11509 1/20 0.42
TSHR P16473 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5352313 0.80 MAPT (0.42) MAPTMAPK1HTTCHRNB2CHRNA4
SCHEMBL27923808 0.78 CHKA (0.46) MAPTNPSR1
SCHEMBL28380433 0.77 LMNA (0.31) MAPTNPSR1
SCHEMBL29626231 0.73 CYP2A6 (0.41) MAPTMAPK1HTTCHRNB2CHRNA4
SCHEMBL27977591 0.73 CYP2A6 (0.41) MAPTMAPK1HTTCHRNB2CHRNA4
SCHEMBL29137307 0.71 CYP2A6 (0.40) MAPTMAPK1HTTCHRNB2CHRNA4
Benzene SCHEMBL28093687 0.71 MAPT (0.41) MAPTMAPK1HTTCHRNB2CHRNA4
SCHEMBL28194545 0.71 CHRNB2 (0.42) MAPTMAPK1HTTCHRNB2CHRNA4
Pyrazole SCHEMBL28821521 0.71 MAPT (0.38) MAPTMAPK1HTTNPSR1
SCHEMBL983193 0.70 CYP2A6 (0.42) MAPTMAPK1HTTCHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020045618-A1 Heteroaryl diazacycloalkanes, their preparation and use NEUROSEARCH A/S (DK) 2002-04-18 US claimed
CN-113999201-B Synthesis and preparation method of nicotine 成昌梅 2023-11-03 CN disclosed
CN-113999201-A Synthetic preparation method of nicotine 成昌梅 2022-02-01 CN disclosed
US-20180042909-A1 Methods of Treating Cancers, Autoimmune Disorders, and Other Conditions Associated with Chronic Inflammation MYMD PHARMACEUTICALS, INC. (US) 2018-02-15 US disclosed
US-20180042909-A1 Methods of Treating Cancers, Autoimmune Disorders, and Other Conditions Associated with Chronic Inflammation MYMD PHARMACEUTICALS, INC. (US) 2018-02-15 US disclosed
CN-106470976-A The method of preparation 3 (3 chlorine 1H pyrazoles 1 base) pyridine 美国陶氏益农公司 2017-03-01 CN disclosed
US-20020045618-A1 Heteroaryl diazacycloalkanes, their preparation and use NEUROSEARCH A/S (DK) 2002-04-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020045618-A1 Heteroaryl diazacycloalkanes, their preparation and use CHRNA5, CHRNA7, CHRNA3 MAPT 1195/4885MAPK1 1592/4885HTT 885/4885
US-20180042909-A1 Methods of Treating Cancers, Autoimmune Disorders, and Other Conditions Associated with Chronic Inflammation ROS1, NOX4, MPO MAPT 1874/4885MAPK1 811/4885HTT 187/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.